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Receptors and effect
Lecture 8
Receptor | Effect |
---|---|
D2 receptor: | Extrapyramidal Syndromes (EPS) |
D2 receptor: | Dystonia |
D2 receptor: | Akathisia |
D2 receptor: | Parkinsonism |
D2 receptor: | Tardive Dyskinesia |
D2 receptor: | Neuroleptic Malignant Syndrowme (NMS) (altered mental status, motor symptoms, hyperthermia, autonomic instability) |
α1-adrenergic receptor: | Hypotension |
H1 receptor: | Increased appetite |
Muscarinic receptor: | Anticholinergic |
Serotonin receptor 5HT2A: | Decreased anxiety Helps with sleep (benefit) |
Fast sodium channel: | Cardiac problems Increased QRS |
GABAA receptor: | Seizures Don't see very often |