click below
click below
Normal Size Small Size show me how
Ax Drugs
Major Types & Reversal Drugs
| Question | Answer |
|---|---|
| Morphine | Full agonist - Opioid |
| Hydromorphone | Full agonist - Opioid 8 X more potent than Morphine |
| Fentanyl | Full agonist - Opioid 75-100X more potent than Morphine |
| Tramadol | Post op full agonist opioid used for pain |
| Buprenorphine | Partial agonist opioid (LONG duration , moderate analgesia) |
| Butorphanol | K Agonist/ Mu Antagonist Opioid SHORT duration, minimal analgesia & sedation |
| Naloxone | Opoid ANTagonist (will reverse both sedation AND analgesia!!) |
| Naltrexone | potent long lasting opioid antagonist |
| Atropine | Anti-cholinergic - inc HR, dec secretions, dec GI motility |
| Glycopyrrolate | Anti-cholinergic - inc HR, dec secretions, dec GI motility - DOESNT CROSS THE BBB |
| Acepromazine | Phenothiazine - SLOW onset of action |
| Diazepam | Benzodiazepine - GABA agonist |
| Midazolam | Benzodiazepine - GABA agonist |
| Flumazenil | GABA ANTAgonist -- reversal for benzodiazepine |
| Xylazine | Alpha-2 agonist |
| Medetomidine | Alpha-2 agonist - much more potent than xylazine (75x) - profound long lasting sedation, analgesia |
| Dexmedatomidine | Alpha-2 agonist |
| Detomidine | Alpha-2 agonist |
| Romifidine | Alpha-2 agonist |
| Ketamine | Dissociative Anesthetic |
| Telazol | Dissociative (Tiletamine) + Zolazepam |