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Pharm Fall 2012
| Question | Answer |
|---|---|
| epinephrine | adrenergic agonist, alpha and beta |
| phenylpropanolamine | adrenergic agonist, alpha and beta |
| dopamine | adrenergic agonist, alpha 1, beta 1 |
| dobutamine | adrenergic agonist, alpha 1, *beta 1*, beta 2 |
| phenylephrine | adrenergic agonist, alpha 1 |
| isoproteronol | adrenergic agonist, beta 1 & beta 2 |
| albuterol | adrenergic agonist, beta 2 |
| clenbuterol | adrenergic agonist, beta 2 |
| carvedilol | adrenergic antagonist, alpha 1, beta 1, beta 2; class II antiarrhythmic |
| phenoxybenzamine | adrenergic antagonist, alpha 1 & 2 |
| propanolol | adrenergic antagonist, beta 1 & 2; class II antiarrhythmic |
| timolol | adrenergic antagonist, beta 1 & 2 |
| atenolol | adrenergic antagonist, beta 1 |
| bethanecol | cholinergic agonist, direct, muscarinic |
| pilocarpine | cholinergic agonist, direct, muscarinic |
| carbachol | cholinergic agonist, direct, muscarinic & nicotinic |
| physostigmine | cholinergic agonist, indirect, muscarinic & nicotinic |
| neostigmine | cholinergic agonist, indirect, muscarinic & nicotinic |
| edrophonium | cholinergic agonist, indirect, muscarinic & nicotinic |
| pyridostigmine | cholinergic agonist, indirect, muscarinic & nicotinic |
| organophosphates | cholinergic agonist, indirect, muscarinic & nicotinic |
| atropine | cholinergic antagonist, muscarinic (decrease secretions/GI motility, increase HR, bronchodilation, decrease bladder contractions) |
| glycopyrrolate | cholinergic antagonist, muscarinic (decrease secretions/GI motility without cardiovascular effect) |
| lidocaine | local anesthetic; amide-linked; class I antiarrhythmic |
| mepivicaine | local anesthetic, amide-linked |
| bupivicaine | local anesthetic, amide-linked |
| benzocaine | local anesthetic, aminoester |
| proparacaine | local anesthetic, aminoester |
| atracurium | neuromuscular blocker; competitive (nondepolarizing) |
| vecuronium | neuromuscular blocker; competitive (nondepolarizing) |
| pancuronium | neuromuscular blocker; competitive (nondepolarizing) |
| succinylcholine | neuromuscular blocker; depolarizing |
| morphine | opioid; mu, kappa |
| hydromorphone | opioid; mu |
| codeine | opioid; mu |
| fentanyl | opioid; mu |
| buprenorophine | opioid; mu |
| butorphanol | opioid; mu, kappa |
| nalbuphine | opioid; mu antagonist, kappa agonist |
| naloxone | opioid; mu, kappa, delta (all antagonist) |
| naltrexone | opioid; mu, kappa, delta (all antagonist) |
| tramadol | opioid; mu, alpha-2; 5-HT (serotonin) [all agonist]; M1 (muscarinic) [antagonist] |
| phenobarbital | anticonvulsant; barbiturate |
| primidone | anticonvulsant; barbiturate |
| phenytoin | anticonvulsant; blocks inward movement of Na+ |
| diazepam | anticonvulsant; anxiolytic (behavior modification); benzodiazepine |
| clonazepam | anticonvulsant; benzodiazepine |
| clorazepate | anticonvulsant; anxiolytic (behavior modification); benzodiazepine |
| felbamate | anticonvulsant; N-methyl D-aspartate antagonist |
| gabapentin | anticonvulsant; blocks Ca2+ channels |
| levetiracetam | anticonvulsant; unknown MoA, possibly binding SV2A = inhibit presynaptic Ca2+ channels |
| zonisamide | anticonvulsant; blocks inward movement of Na+ |
| potassium bromide | anticonvulsant; unknown MoA; changes K+ influx |
| buspirone | behavior modification (anxiolytic); azapirone |
| amitriptyline | behavior modification; tricyclic antidepressant |
| clomipramine | behavior modification; tricyclic antidepressant |
| fluoxetine | behavior modification; selective serotonin reuptake inhibitor |
| paroxetine | behavior modification; selective serotonin reuptake inhibitor |
| selegiline | behavior modification; monoamine oxidase type B inhibitor |
| midazolam | benzodiazepine |
| lorazepam | benzodiazepine |
| flumazenil | benzodiazepine antagonist (competitive) |
| acetazolamide | diuretic - carbonic anhydrase inhibitor |
| mannitol | diuretic - osmotic diuretic |
| furosemide | diuretic - loop diuretic |
| chlorothiazide | diuretic - thiazide diuretic |
| hydrochlorothiazide | diuretic - thiazide diuretic |
| triamterine | diuretic - inhibitor of renal epithelial sodium channels |
| amiloride | diuretic - inhibitor of renal epithelial sodium hcannels |
| spironolactone | diuretic - antagonist of mineralocorticoid receptors |
| ammonium chloride | urinary tract drug - urine acidifier |
| dantrolene | urinary tract drug - relax urethra (cats) |
| potassium citrate | urinary tract drug - alkalinizes urine |
| digoxin | positive inotrope: inhibits Na-K-ATPase |
| pimobendan | inodilator (+ inotrope, vasodilator): inhibits phosphodiesterase III |
| diltiazem | vasodilator (Ca channel blocker = decrease intracellular Ca2+); class IV antiarrhythmic |
| amlodipine | vasodilator (Ca channel blocker = decrease intracellular Ca2+) |
| hydralazine HCl | vasodilator (direct arteriolar dilator) |
| enalapril | ACE inhibitor |
| benazepril | ACE inhibitor |
| quinidine | class I antiarrhythmic |
| procainamide | class I antiarrhythmic |
| amiodarone | class III antiarrhythmic |
| sotalol | class III antiarrhythmic |
| virapamil | class IV antiarrhythmic |