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Block 3 Drugs
| Question | Answer |
|---|---|
| Cimetidine trade name | Tagamet |
| Cimetidine class | H2 antag |
| Ranitidine trade name | Zantac |
| Ranitidine class | H2 antag |
| Famotidine trade name | Pepcid |
| Famotidine class | H2 antag |
| Omeprazole trade name | Prilosec |
| Omeprazole class | Proton pump inhibitor |
| Metronidazole class | Nitroimidazol antibiotic |
| Amoxicillin class | Penicillin antibiotic |
| Clarithomycin class | Macrolide antibiotic |
| AlOH3 and MgOH2 trade name | Mylanta, Maalox |
| Mylanta, Maalox class | Antacid Salt |
| Calcium Carbonate trade name | Tums |
| Tums class | Antacid Salt |
| Sodium Bicarbonate trade name | Alka Seltzer |
| Alka Seltzer class | Antacid Salt |
| Sucralfate trade name | Carafate |
| Sucralfate class | Mucosal protective agent |
| Misoprostol trade name | Cytotec |
| Misoprostol class | Mucosal Protective Agent |
| Bismuth Subasalicylate trade name | Pepto Bismol |
| Bismuth Subsalicylate class | Mucosal Protective Agent |
| Metoclopramide trade name | Reglan |
| Metoclopramide class | Prokinetic Agent |
| Cimetadine Adverse | blocks P450s |
| Famotidine Advantage | does not inhibit first pass ethanol metabolism |
| Proton Pump Inhibitor MOA | covalent modification of H/K ATPase- irreversible |
| Zollinger-Ellison treatment of choice | Proton Pump Inhibitors |
| Sucralfate MOA | produces protective covering of ulceration |
| Misoprostol MOA | Prostaglandin receptor agonist- inc. secretion of mucous and bicarb |
| Misoprostol Adverse | causes myometrial contrxn- no use in pregnancy |
| Metoclopramide MOA | 5-HT4 receptor agonist- gastric emptying |
| Ciprofloxacin trade name | Cipro |
| Ciprofloxacin class | Fluorinated 4-quinolone |
| Ofloxacin trade name | Floxin |
| Ofloxacin class | Fluorinated 4-quinolone |
| Norfloxacin class | Fluorinated 4-quinolone |
| Octreotide trade name | Sandostatin |
| Octreotide class | Somatostatin analog |
| Diphenoxylate trade name | Lomotil |
| Diphenoxylate class | Piperidine opioid mu agonist |
| Difenoxin trade name | Motofen |
| Difenoxin class | Piperidine opioid mu agonist |
| Loperamide trade name | Imodium |
| Loperamide class | Piperidine opioid mu agonist |
| Ondensatron trade name | Zofran |
| Ondensatron class | 5-HT3 Antagonist |
| Granisetron trade name | Kytril |
| Granisetron class | 5-HT3 Antagonist |
| Trimethobenzamide trade name | Tigan |
| Trimethobenzamide class | D2 antagonist- prokinetic agent |
| Chlorpromazine trade name | Thorazine |
| Chlorpromazine class | Neuroleptic |
| Prochlorperazine trade name | Compazine |
| Prochlorperazine class | Neuroleptic |
| Heloperidol trade name | Haldol |
| Heloperidol class | Neuroleptic |
| Dexamethasone class | Glucocorticoid |
| Dronabinol trade name | Marinol (pot) |
| Dronabinol class | Cannabinoid |
| Lorazepam trade name | Ativan |
| Lorazepam class | Benzodiazepines |
| Promethazine class | Antihistamine |
| Scopolamine class | Anticholinergic |
| Ipecac | Emetic |
| Opioid MOA | Reduced motility, acid- antidiarrheal |
| Fluorinated 4- quinolones MOA | Inhibit A subunit of DNA gyrase |
| Bismuth salicylate MOA | coating ulceration (dyspepsia), antimicrobial(ulcers and diarrhea) |
| mu opioid agonists MOA | inhib of presynaptic nerves of myenteric plexus- low motility |
| Difenoxylate, Difenoxin Adverse | Affect CNA- can be addictive |
| Octreotide MOA | Interaction with somatostatin receptor |
| Octreotide Adverse | gallstones due to decreased emptying |
| 5-HT3 receptor antagonists MOA | block 5-HT3 receptor- anti-emetics |
| Metoclopramide anti-emetic MOA | 5-HT3 agonist, D2 antag- inc. motility |
| Dexamethasone MOA | decrease inflammation- anti-emetic |
| Dronabinol MOA | Cannabinoid agonist- anti-emetic |
| Promethazine, Diphenylhydramine MOA | H1 receptor antagonists- motion sickness and vertigo |
| Scopolamine MOA | Muscarinic antagonist- motion sickness |
| Apomorphine class | pro-emetic (poisoning)- stimulates the CTZ |
| Diuretics | Compounds that produce salt excretion |
| Diuretic uses | CHF, Hypertension, Edema |
| Acetazolamide trade name | Diamox |
| Acetazolamide class | CA inhibitor |
| Dichlorophenamide trade name | Daranide |
| Dichlorophenamide class | CA inhibitor |
| Methazolamide trade name | Neptazane |
| Methazolamide class | CA inhibitor |
| CA inhibitor uses | Glaucoma, Cerebral Edema, Alkalosis |
| CA inhibitor MOA | dec. reabs. of bicarb |
| Glycerin class | Osmotic Diuretic |
| Isosorbide class | Osmotic Diuretic |
| Mannitol class | Osmotic Diuretic |
| Urea class | Osmotic Diuretic |
| Osmotic Diuretic MOA | osmotically keep water in tubule- excretion |
| Ethacrynic Acid trade name | Edecrin |
| Ethacrynic Acid class | Loop Diuretic |
| Furosemide trade name | Lasix |
| Furosemide class | Loop Diuretic |
| Bumetanide trade name | Bumex |
| Bumetanide class | Loop Diuretic |
| Torsemide trade name | Demadex |
| Torsemide class | Loop Diuretic |
| Loop Diuretic MOA | look up! |
| Loop Diuretic secretion | not filtered- secreted in prox tubule |
| Loop Diuretic adverse | K+ wasting, hyponatremia |
| Chlorothiazide trade name | Diuril |
| Chlorothiazide class | Thiazide diuretic |
| Hydrochlorothiazide trade name | Hydrodiuril |
| Hydrochlorothiazide class | Thiazide diuretic |
| Thiazide MOA | Inhib NaCl symport in dist tubule |
| Thiazide adverse | tolerance after 1 wk, lethal with Quinidine (antiarrhythmetic) |
| Amiloride trade name | Midamor |
| Triamterene trade name | Dyrenium, Maxide |
| Amiloride class | Na+ channel inhibitor |
| Triamterene class | Na+ channel inhibitor |
| Na+ channel inhib advantage | K+ sparing |
| Na+ channel inhib MOA | Inhib Na+ channel in dist tubule |
| Spironolactone trade name | Aldactone |
| Spironolactone class | Aldosterone Antagonist |
| Aldosterone Antagonist MOA | Prevents ALDO-MR binding, dec. Na+ reabs and K+ secretion |
| T. enanthate, cypionate, propionate | IM Testosterone replacements |
| Testoderm | Transcrotal Testosterone replacement |
| Androderm | Transdermal Testosterone replacement patch |
| Androgel | Transdermal Testosterone replacement gel |
| Testopel | subQ implant testosterone replacement |
| Sildenafil trade name | Viagra |
| Sildenafil MOA | PDE 5 inhibitor- inc. cGMP, vasodilation |
| Sildenafil use | Tx. of ED |
| Vardenafil trade name | Levitra |
| Vardenafil MOA | PDE 5 inhibitor- inc. cGMP, vasodilation |
| Vardenafil use | Tx. of ED |
| Tadalafil trade name | Cialis |
| Tadalafil MOA | PDE 5 inhibitor- inc. cGMP, vasodilation |
| Tadalafil use | Tx. ED |
| Yohimbine class | a2 adrenergic antagonist |
| Yohimbine use | Tx. psychogenic ED |
| Papaverine | opioid peptide |
| Papaverine | injected tx. for ED |
| Phentolamine | alpha adrenergic antag |
| Phentolamine | injected tx. for ED |
| Alprostadil class | PGE1 |
| Alprostadil admin route | penile injection or urethral pellet |
| Alprostadil use | Tx. ED |