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MEDS 301
Intro to Pharmacology
| Question | Answer |
|---|---|
| Aptamer | Pegaptanib |
| Fusion Protein | Etanercept |
| MAB | Bevacizumab |
| Antisense | Oblimersen |
| Antibiotic: Cell Wall Inhibitor | Penicillin |
| Antibiotic: 50S Ribosomal Inhibitor | Macrolides (Erythromycin) |
| Antibiotic: 30S Ribosomal Inhibitor | Tetracycline Aminoglycosides |
| Antibiotic: RNA Polymerase Inhibitor | Rifamycin |
| Antibiotic: DNA Gyrase Inhibitor | Fluoroquinolones (Ciprofloxacin) |
| Antibiotic: Purine Synthesis Inhibitor | Trimethoprim/Sulfamethoxazole |
| Antifungal: Cell Wall Inhibitor | Echinocandins (Caspofungin) |
| Antifungal: Cell Membrane Inhibitor | Polyenes (Nystatin) Allylamines (Terbinafine) Clotrimazole |
| Antiviral: Attachment CCR5 Inhibitor | Maraviroc |
| Antiviral:DNA Polymerase Inhibitor | Acyclovir |
| Antiviral: RNA Reverse Transcriptase Inhibitor - nucleoside | Zidovudine |
| Antiviral: RNA Reverse Transcriptase Inhibitor - non nucleoside | nevirapine |
| Antiviral: Uncoating proton channel inhibitor | Amantadine |
| Antiviral: Integrase Inhibitor | Raltegravir |
| Antiviral: Maturase Protease Inhibitor | Ritonavir |
| Antiviral:Release Neuraminidase Inhibitor | Oseltamavir |
| Cancer: DNA Damaging | Alkylating agents, Platinum, Anti-tumor antibiotics |
| Cancer: Anti-tumor antibiotics | Belomycin |
| Cancer: DNA synthesis/repair inhibitors - nonmetabolites | Folate analogues (methotrexate) Purine analogues (Mercaptopurine) Pyrimidine analogues (Fluorouracil) |
| Cancer: DNA synthesis/repair inhibitors - topoisomerase inhibitors | Anthracyclines (Doxorubin) |
| Cancer: Microtubule Inhibitors | Taxanes Vinca Alkaloids |
| CADS: Growth Factor Inhibitors | ERGF: gefitinib BCR-ABL: imantinib HER-2: Trastuzumab |
| CADS: Angiogenesis Inhibitor | VEGF: Bevacizumab |
| CADS: Anti-Apoptosis Inhibitor | Oblimersen |
| Sympatholytics | Beta receptor blockers: propranolol Decrease NT: clonidine |
| Acetylcholine Inhibitor | Atropine |
| Antihypertensive: Diuretics | Thiazides: Hydrochlorothiazide Loop Diuretics: Furosemide K+ Sparing: Spirinolactone |
| Antihypertensive: ACE Inhibitors | captopril |
| Antihypertensive: Angiotension Receptor Blocker | Losartan |
| Antihypertensive: Renin Inhibitor | aliskeren |
| Antihypertensive: Calcium channel blocker - dihydropyridine | nefidipine |
| Antihypertensive: Calcium channel blocker - non dihydropyridine | benzothiazepine (diltiazem) phenylalylamine (verapamil) |
| Antihypertensive: Beta blockers - cardioselective | atenolol |
| Antihypertensive: Beta blockers - non cardioselective | propranolol carvedilol |
| Antihypertensive: Beta blockers - partial agonist | Acebutolol |
| Antihypertensive: alpha 1 antagonist | prazosin |
| Antihypertensive: vasodilators | hydralazine |
| Antihypertensive: alpha 2 agonist | clonidine |
| Antihypertensive: endothelin antagonist | bosentan |
| Antihypertensive: vasopeptidase inhibitors | omepatrilat |
| Heart Failure: Help heart pump efficiently | Digitalis Glycosides (Digoxin) |
| Heart Failure: Reduce resistance | ACE inhibitors |
| Heart Failure: reduce work | Beta blockers |
| Stable Angina: Reduce Oxygen Demand | Beta blockers Nitrates (nitroglycerin) Calcium channel blockers (non-dihydropyridines) |
| Variant Angina: relieve muscle spasm | Calcium channel blockers (dihydropuridines) Nitrates |
| Treat Heart Attacks | Statins (Atorvastatin) |