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physio drugs
Term | Definition |
---|---|
Botulismtoxin | Prevents release of ACh from vesicle. Degrades Synaptobrevin. |
Neostigmine | Reversible AChE Inhibitor |
Physostigmine | Reversible AChE inhibitor. Crosses BBB |
Edrophonium | Reversible AChE inhibitor. |
Parathion | Irreversible AChE inhibitor |
Succinylcholine | Neuromuscular Nicotinic Agonist |
Pancuronium | Neuromuscular Nicotininc Antagonist. used in surgery |
Acetylcholine | Muscarinic agonist |
Pilocarpine | Muscarinic agonist. used for glaucoma |
Methacholine | Muscarinic agonist |
bethanechol | Muscarinic agonist. used for post op GI motility |
Atropine | muscarinic antagonist. Bind muscarinic receptors to block them |
Amphetamine | Inhibits Catecholamine storage |
Pseudophedrine | Inhibits Catecholamine storage |
Cocaine | Inhibits Catecholamine reuptake |
imipramine | Inhibits Catecholamine reuptake |
Iproniazid | Inhibits Catecholamine metabolism |
Epinephrine | Alpha & Beta Agonist |
Norepinephrine | Alpha & Beta Agonist |
Oxymetazoline | Alpha 1 & Alpha 2 Agonist |
Phenylephrine | Alpha 1 Agonist |
Clonidine | Alpha 2 agonist |
Phenoxybenzamine | Alpha 1 & Alpha 2 antagonist. used to treat pheochromocytoma |
Phentolamine | Alpha 1 & Alpha 2 antagonist |
Prazosin | Alpha 1 antagonist |
Tamsulosin | Alpha 1 antagonist |
Dobutamine | Beta 1 Agonist |
Albuterol | Beta 2 agonist |
Propanolol | Non-selective Beta blocker. Contraindicated in asthma patients |
Atenolol | Selective Beta 1 blocker |
Pindolol | Partial Agonist |