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Antianginal Drugs
Drugs recognition: chap 11
| Question | Answer |
|---|---|
| isosorbide dinitrate (Isordil) | Organic Nitrates |
| isosorbide mononitrate (Imdur) | Organic Nitrates |
| nitroglycerin (sl tabs, sl sprays, topical…) | Organic Nitrates |
| amlodipine (Norvasc) | Calcium Channel Blockers/Dihydropyridines |
| felodipine (Plendil) | Calcium Channel Blockers/Dihydropyridines |
| nifedipine (Procardia, Adalat) | Calcium Channel Blockers/Dihydropyridines |
| nicardipine (Cardene) | Calcium Channel Blockers/Dihydropyridines |
| diltiazem (Cardizem, Diltia) | Calcium Channel Blockers/Non-dihydropyridines |
| verapamil (Verelan, Calan) | Calcium Channel Blockers/Non-dihydropyridines |
| atenolol (Tenormin) | Beta Blockers |
| metoprolol (Lopressor, Toprol XL) | Beta Blockers |
| propranolol (Inderal) | Beta Blockers |
| nadolol (Corgard) | Beta Blockers |
| Ranolazine (Ranexa) | Metabolic Modifier |
| nitroglycerine (organic nitrates) | Acute angina & cyanide poisoning multiple routes of administration |
| nitroglycerine Adverse effects | HA, hypotension, reflex tachy |
| calcium channel blockers (-ine, verapamil, diltiazem) adverse effects | Peripheral edema, gingival hyperplasia |
| calcium channel blockers moa | Smooth muscle relaxation & suppress cardiac activity, Reduce heart rate & contractility |
| atenolol (Tenormin) propranolol (Inderal) indications | Prevent ischemic episodes & reflex tachycardia Post-MI – improve survival & decrease risk of recurrence |
| ranolazine (Ranexa) | No decrease in BP or HR Increase exercise capacity & reduce angina Increased efficiency of glucose metabolism Generates more energy per oxygen used |
| nitroglycerine | cant take with viagra |