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tara's pharm part 2 final review

Quiz yourself by thinking what should be in each of the black spaces below before clicking on it to display the answer.
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Question
Answer
pt on 5th day vanco and gent, tv is really loud   show
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show (A) NOT ORALLY ABSORBED (E) RENAL EXCRETION-IF DECREASE RENAL FUNCTION-LONGER DOSING INTERVAL  
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show CELL WALL LYTIC-COVERS GRAM + ONLY (MRSA, C-DIFF)  
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show IF TOXIC-RISK FOR NEPHRO/OTO TOXICITY-SO IT CAN AFFECT IT'S OWN HALF LIFE IN TOXIC DOSES, REDMAN SYNDROME-SYSTEMIC WILL CAUSE HIVES, HYPOTENSION  
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show SHOULD BE SLOWER INFUSION RATE  
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VANCO (PK)   show
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show PREVENT PROTEIN SYNTHESIS, COVERS GRAM - ONLY,EXCEPT WHEN ADDED TO TO BETA-LACTAMS OR VANCO B/C RIBOSOME IS INSIDE CELL AND THOSE BETA-LACTAMS AND VANCO CAN BREAK CELL WALL-COMBO=SYNERGY(1+1=3)  
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show THESE DRUGS HAVE THERAPEUTIC WINDOWS AS WELL,SO NEED PEAKS AND TROUGHS, NOT ORALLY ABORSBED, iV ONLY,HALF LIFE UPON RENAL FUNCTION  
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S/E RIBOSOMALS   show
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MACROLIDES-ERYTHROMYCIN EX;CLARITHROMYCIN, AZITHROMYCIN(Z-PACK) (PD)   show
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show ALL ARE POTENT (METABOLIC ENZYME INHIBITORS) SO AVOID OTHER DRUGS W/ THERAPEUTIC WINDOW B/C IT WILL INCREASE OTHER DRUGS AFTER TIME (TOXICITY)  
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AZITHROMYCIN (PK)   show
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CLIENT HAD 10 DAYS THERAPY OF ABX-FAILED AND WANTS TO KNOW WHY Z-PACK IS ONLY COUPLE DAYS   show
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show METALLIC TASTE ALL CHEMICAL SIMILAR TO GUT...DIARRHEA  
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SULFONAMIDES-BACTRIM SEPTRA(AVOID SUN) (PD)   show
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SULFONAMIDES (PK)   show
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SULFONAMIDES S/E   show
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show DO OPPOSITE OF PCN AND CEPHS, EARLY;CIPRO G- > + , NEWER;LEVAQUIN G+ = -  
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show CAN INHIBIT CAFFEINE AND THEOPHYLLINE METABOLISM  
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QUINOLONES S/E   show
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TUBERCULOSIS-ACID FAST MYCOBACTERIA   show
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show DRUGS CAN MAKE YOU FEEL WORSE THEN THE DX THEREFORE COMPLIANCE IS PROBLEM, ALL REGIMENS ARE HEPATOTOXIC TO SOME DEGREE-S/S YELLOWING OF SKIN/EYES, ASH COLORED STOOLS-AVOID ALCOHOL AND ACETAMINOPHEN  
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show 1)RIFAMPIN-CAUSES RED/ORANGE STAINING OF URINE AND TEARS 2) ISONIAZID (INH)-CAN CAUSE PERIPHERAL NEUROPATHY-TINGLING/NUMBNESS OF FINGERS/TOES-SO ADD VIT B6/PYRIDOXINE  
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show ETHAMBUTOL/MYAMBUTOL-CAN CAUSE TRANSIENT RED/GREEN COLOR BLINDNESS-DON'T DRIVE  
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show ACT LIKE BETA-LACTAMS ON FUNGAL YEAST CELL WALLS AND MEMBRANES  
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ANTIFUNGAL (PK)   show
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show WEAKEST-KETOOCONAZOLE/NIZORAL....FLUCONAZOLE/DIFLUCAN...STRONGEST- ITRACONAZOLE/SPORONOX....SHOULD START W/ THE WEAKEST HOWEVER KETOCONAZOLE NEEDS AN ACIDIC ENVIRONMENT TO BE ABSORBED  
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CLIENT FAILS ON ONE WEEK NIZORAL   show
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show INHIBIT vdna replication(failed chemotherapy agents)  
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antivirals s/e   show
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ganciclovir   show
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show UNINHIBITED CAN MEK 5 BILLION COPIES IN 24 HOURS- 80%NORM/NULL 19% FATAL MUTATION <1% BENEFICIAL TO VIRUS MUTATION -SO TAKE DRUGS ON TIME TO PREVENT 1% MUTATION EX 3X/DAY= Q8HOURS(IMPORTANT)  
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TX OF SHOCK-DECREASED BP=DECREASED PERFUSION   show
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ALPHA EX;TETRAHYDRALOZINE   show
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BETA 1   show
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show BRONCHODILATOR (LUNGS)  
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EPINEPHRINE   show
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NOREPINEPHRINE   show
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show SNS AGONIST ^BP TITRATEABLE=DIFFERENT DOSES DO DIFFERENT THINGS  
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show LOW DOSE-AGONIST AT DOPAMINE RECEPTOR IN THE SPLANCHIC BEDS.. RENAL DOSE(VASODILATOR)..... MED DOSE-BETA 1 AGONIST=^HR,^STRENGTH (CARDIAC)... HIGH DOSE=BETA 1 AND ALPHA AGONIST  
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DOBUTAMINE ^BP   show
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^ STRENGTH OF HEART   show
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show NEGATIVE INOTROPIC EFFECT  
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^HR   show
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DECREASED HR   show
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show VESSELS-CONSTRICT FAST.. .KIDNEYS- RETAIN FLUID (SLOW)  
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show (PK) SNS ANTAGONIST, BETA 1 AND BETA 2, WILL HAVE NEGATIVE CHRONOTROPIC AND INOTROPIC EFFECTS  
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show FLAT AFFECT, NIGHTMARES  
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show ASTHMA (IF IT ENDS IN -OLOL IT BLOCKS DILATION) AND TREATED DIABETES (MASKS THE S/S OF HYPOGLYCEMIA  
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show (PD) NEG CHRONO/INOTROPIC- MAKES CA LESS AVAILABLE FOR MYOCARDIAL CONTRACTIONS AND SLOWS IMPULSE CONDUCTION-IF SOMEONE IS DX W/ DIABETES 2, YOU CAN SWITCHED THE PERSON TO THIS DRUG  
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show (PO) CONSTIPATION  
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COMPENSATORY FOR VASODILATORS (DECREASE BP)   show
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ALPHA BLOCKERS (-ZOSIN) EX TERAZOSIN/HYTRIN   show
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show 1ST DOSE EFFECT-ORTHOSTATIC HYPOTENSION-TAKE AT BEDTIME TO PREVENT INJURY  
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NEW CA CHANNEL BLOCKERS (-DIPINE) EX; DIFEDIPINE/PROCARDIA   show
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show ORTHOSTATIC HYPOTENSION, CONSTIPATION-STAY HYDRATED, MILD EDEMA  
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show DRY COUGH ORTHOSTATIC HYPOTENSION MILD EDEMA POTASSIUM RETENTION MORE IN ELDERLY  
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ANGIOTENSION 2 RECEPTOR BLOCKERS "SARTAN" EX; VALSARTAN/DIOVAN S/E   show
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show WORKS ON KIDNEYS (PD) WHERE SALT GOES WATER FOLLOWS  
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show STRONGEST-LOOP DIURETICS; FURESIMIDE/LASIX (LAST 6 HOURS)-LOSE ALOT OF ELECTROLYTES AVAIL PO/IV....THIAZIDES;CHLORTHALIDONE/HYGROTON DO RETAIN CALCIUM...K+ SPARING;SPIROMALACTONE/ALDACTONE-LOSE NA RETAIN K+-RETENTION WILL INCREASE WITH AGE  
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CLIENT NEEDS FLUID LOSS NOW GIVE   show
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show ARE SULFA RELATED  
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show ELECTROLYTE PANELS-LOOP/THIAZIDE= GREATEST RISK FOR ELECTROLYTE IMBALANCE  
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COMPENSATORY FOR DIURETICS   show
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CAD/ANGINA   show
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NEW CA+ CHANNEL BLOCKERS AND ACE INHIBITORS   show
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BETA BLOCKERS AND OLD CA+ CHANNEL BLOCKERS   show
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show TX;NITROGLYCERIN SL OR BUCCAL SPRAY-DECREASES DIASTOLIC UP TO 40 MMHG  
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show MASSIVELY POTENT VASODILATOR-^O2 SUPPLY (MICRO) AND DECREASES O2 DEMAND (MACRO)  
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show NEED TO BE SITTING DOWN, GOOD UNTIL EXPIRATION HOWEVER, KEEP EXTRA UNOPENED BOTTLE HANDY, IF IT'S GOOD IT WILL TINGLE-CHECK POLICY-TAKE ONE Q 5MIN TIMES 3-CALL 911 AFTER 3RD DOSE-DON'T KEEP IN GLOVE BOX OF CAR  
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show UNDER TONGUE-IF SWALLOWED HAS A LARGE 1ST PASS EFFECT-WHICH MEANS NO DRUG WILL GET IN BODY HALF LIFE AROUND 1 MIN  
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NTG PATCH   show
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CHF   show
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EARLY/LATE TX OF CHF   show
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show SLOWS AND STRENGTHENS THE HEART, NEG CHRONATROPIC, POSITIVE INOTROPIC TO IMPORVE HEART EFFICIENCY-INHIBITS NA/K+ PUMP, SHUTS ELECTROLYTES AWAY FROM NA/K+ AND TOWARD CALCIUM(WHICH ALL SLOWS HEART AND INCREASES STRENGTH)  
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DIGOXIN   show
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show (A)-PO TABLET...NO (D)..NO (M)..(E)-GOES STRAIGHT TO RENAL EXCRETION SO B4 START NEED TO KNOW RENAL FUNCTION (BUN/CREAT)  
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show ^BUN/CREAT=LONGER HALF LIFE, HALF LIFE TAKES ABOUT 24 HOURS W/ NORMAL RENAL FUNCTION, WHEN STARTING IT TAKES A LIL TIME TO BUILD UP TO THERAPEUTIC (2-3 DAYS) B/C THERAPEUTIC WINDOW  
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DIGOXIN   show
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DIGOXIN   show
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show ^ OR DECREASE K+= ^DIG TOXICITY  
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DIGOXIN S/S TOXICITY (PT)   show
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show BY MEDIC ALERT BRACLET, WEEKLY PILL ORGANIZER, KEEP TRACK OF NA, IF YOU LOSE DOPPLER GET ANOTHER ONE( CHILD)  
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DIGOXIN ANTIDOTE-DIGOXIN IMMUNE FAB/DIGIBIND   show
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show CLASS 1=SODIUM CHANNEL BLOCKERS.. .CLASS 2= BETA BLOCKERS... CLASS 3= AMIODARONE/CORDARONE (BEST ONE)  
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show CAN CHANGE TO OLD CA+ CHANNEL BLOCKERS AKA CLASS 4  
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ANTIARRHYTHMICS (PK)   show
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BETA BLOCKERS CAN BE TAKEN FOR MANY REASONS   show
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show NEGATIVE CHRONOTROPIC NEGATIVE INOTROPIC  
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show (M) IS SUBJECT TO ENZYME INDUCTION/INHIBITION HALF LIFE;LOADING DOSE PHASE; SHORT HALF LIFE... MAINTENENCE;HALF LIFE ABOUT 35 DAYS=ADR COULD LAST LONG TIME  
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show ORTHOSTATIC HYPOTENSION "RISE SLOWLY", ALTERED THYROID FUNCTION "NEED BASELINE/FOLLOW UP", RARE-RETINAL DEPOSITS(D/C DRUG-COULD LEAD TO BLINDNESS)"IF ANY EYE SIGHT C/O CALL MD, PULMONARY FIBROSIS (SPIROMETRY-BASELINE/FOLLOW UP) AND BLUE/GRAY DISCOLORATION  
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show PULMONARY FIBROSIS  
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show NEED DRUG LEVEL AND THYRIOD PANEL  
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show IF IN ARTERIAL=PLATELTS W/ FIBRIN, VENOUS=FIBRIN W/ PLATELTS EX HEPARIN PREVENTS CLOT FORMATION AND OR EXISTING CLOT GROWTH  
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show PREVENT PLATELET ACTIVATION EX ASPIRIN OR PLAVIZ  
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ANTICOAGULANTS INPATIENT   show
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show WARFARIN/COUMADIN DAGIBACTRAN/PRADAXA  
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show (PD) INHIBITS COAGULATION FACTOR 10 (PK) SHORT HALF LIFE, SO CONTROLLABLE LAB=PTT  
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show HETEROGENOUS MIXTURE- ABSORPTION VARIES FROM BATCH TO BATCH D/T SIZE AND ACTIVITY USE PTT AS A CHECK  
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ENOXAPORIN/LOVENOX (PK)   show
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show LOVENOX  
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show RED/ORANGE TINGE URINE, BLK TARRY/BLOODY STOOL-INSPECT URINE/STOOL DAILY & SKIN DAILY- UNEXPLAINABLE BRUISES-CALL MD...GET FAMILY INVOLVED-MENTAL STATUS CHG..USE ELECTRIC RAZORS, CLOSED TOE SHOES, SLIP/FALL PROFF HOME,NO ALCOHOL, SOFT BRISTLE TOOTHBRUSH  
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show DEFECTIVE FORM OF VIT K, LEADS TO FORMATION OF DEFECTIVE VIT-K DEPENDENT CLOTTING FACTORS- LESS CONTROLLABLE THEN HEPARIN  
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ON DAY 4 OF COUMADIN 2.8 INR WHAT WOULD IT BE BY DAY 8   show
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WARFARIN AND VIT K (FAT SOLUBLE)-CAN STORE IN LIVER   show
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show SPINACH BROCCOLI CAULIFLOWER CABBAGE BRUSSEL SPROUTS KALE... ASPARAGUS(MOST VIT-K) AVOID EXCESS CONSUPMTION  
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PT IS ON WARFARIN THEIR DIET SHOULD BE   show
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show RULE- ASSUME ALL DRUGS INTERACT W/ WARFARIN THEREFORE NEED OF ALL DRUGS LIST AND CHANGE OF DOSES TO BE REPORTED TO MD  
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show BISMUTH SUBSALICYLATE/PEPTO BISMAL METHYL SALICYLATE. OIL OF WINTERGREEN AND ASPERCREAM.. .ALL NEED TO BE AVOIDED WHEN ON WARFARIN B/C IT WILL ^ BLEEDING  
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show PREVENTS PLATELETS ACTIVATION  
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show PREVENTS PROSTOGLANDINS SYNTHESIS.. IS TITRATABLE  
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CLOPIDOGRE/PLAVIX (PD)   show
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ASA WORKS MORE ON STUFF   show
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ASA   show
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show INHIBITS PROSTAGLANDIN SYNTHESIS.. YES-TITRATABLE.. 81MG DOSE- PRIMARY PREVENTION  
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show (PK) KNOWN AS A PRODRUG (IT NEEDS HEPATIC METABOLISM (ONCE TO BE ACTIVATED.. IF YOU INHIBIT (M) IT WON'T BE ACTIVATED..ACTIVATION IS INHIBITED BY PRILOSEC..SLIGHTLY STRONGER THEN ASA  
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PLAVIX   show
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TX OF HIGH CHOLESTEROL   show
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show (PD) INHIBIT HEPATIC CHOLESTEROL SYNTHESIS.. CHOLESTEROL BINDING RESINS- SHOULD TAKE W/ MEALS, TAKE OTHER MEDS -+2 HOURS  
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show HAVE LONG HALF LIFE, STRONGEST ONES  
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STATINS S/E   show
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ASTHMA; PAROXYSMAL BRONCHIAL CONSTRICTION AND INFLAMMATION   show
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show ALBUTEROL ACUTE...STEROID PREVENTATIVE  
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show B2 AGONIST (THERAPEUTIC) AND B1 AGONISTS (^HR ^BP)..SNS AGONISTS  
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show BLACK BOX WARNING  
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CLIENT ADMITS TO OVERUSE OF OF MAINTENENCE INHALER EXPECT TO SEE   show
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STEROID INHALERS BECLOMETHASONE LONG ONSET LONG DURATION S/E   show
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show MORE COMMONLY USED W/ COPD BUT STILL FOR ASTHMA EX IPOTROPIUM/STROVENT TIOTROPIUM/SPIREVA  
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show MAKE B2 AGONIST WORK BETTER  
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show TELL TO HOLD BREATH FOR AS LONG AS COMFORTABLE WHEN INHALING S/E-DRY MOUTH  
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TYPE 2 DIABETES   show
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OLD SCHOOL HYPOGLYCEMIC DRUGS   show
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NEW SCHOOL DIABTETIC MEDS   show
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show W/ TYPE 2 DIABETES HAVE TO TREAT INSULIN AND GLUCAGON-SULFANYLUREAS ADDRESS INSULIN  
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show OLD SCHOOL  
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show TENDS TO NORMALIZE BLOOD SUGAR, SAFER DRUG, COMMONLY 1ST DRUG NEW TYPE 2 DIABETES PUT ON  
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(PD) METFORMIN/GLUCOPHAGE   show
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show C/O SWEATING, CONFUSED=HYPO= GLIPIZIDE CAUSING IT  
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show METFORMIN  
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show 24-48 HOURS PRIOR TO MAJOR SURGERY AND/OR IODINE DYE STUDIES OR IF RENAL IMPAIRED-IF YOU DON'T CAN CAUSE LACTIC ACIDOSIS (RIGIDITY/PAIN ABD.)  
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EPILEPSY-KINDLING THERAPY   show
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EPILEPSY   show
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show PHENTOIN/PHT/DILANTIN... CARBAMAZEPINE/CBZ/TEGRETOL... PHENOBARBITAL/LUMINOL.. VALPORIC ACID/DEPOKOTE..ADD ON(ADJUNCT)- GABAPENTIN/NEURONTIN (S/E SEDATION)  
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WHICH MED FOR EPILEPSY NEEDS TO BE COMBINED W/ OTHER MED   show
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EPILEPSY MED ON BLOOD   show
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IF CLIENT EXPLAINS OF MORE SEIZURES   show
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show ALL PRIMARY MEDS HAVE A RISK OF FOLATE DEFIENCY ANEMIA (TIRED UPON EXERTION)- DISCUSS FOLATE SUPPL W/ MD..RARE-APLASTIC ANEMIA-IF ANY UNUSUAL BRUISING-REPORT TO MD NOW! IF FLU-LIKE S/S OR SORE THROAT-CALL MD  
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show ALL EPILEPSY MEDS HAVE A RISK OF LIVER DAMAGE S/S JAUNDICE AND ASHTON COLORED STOOLS AVOID ETOH AND APAP...HEART=TOXICITY-ALTER HR AND RHYTHM  
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show ENZYME INDUCERS (DECREASE THE LEVEL OF OTHER DRUGS)  
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show ENZYME INHIBITOR (INCREASE LEVELS OF OTHER DRUGS)- THEREFORE TELL MD OF ALL MEDS BEING TAKEN  
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show ALL MEDS CAN CAUSE PHOTOSENSITIVITY "WEAR SUNSCREEN" ALL CAN CAUSE RASHES, IT IS COMMON FOR THEM TO CAUSE A SELF-LIMITING RASH (DOESN'T LAST LONG)... RARE-STEVEN JOHNSONS SYNDROME- USUALLY OCCURS 1ST 6 MONTHS OF STARTING-PROGRESSING- CALL MD  
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show (PK) ZERO ORDER KINETICS HALF LIFE HAS NO MEANING, SO ONLY WAY TO FIND OUT IS TO TAKE LEVEL, SMALL CHANGES IN DOSE CAN CAUSE LARGE CHANGES IN CP-KEEP OUT OF REACH OF CHILDREN  
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PHENYTOIN/DILANTIN S/E   show
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OPIATES S/E   show
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show PHYSICAL- LONG TERM WILL NEED HIGHER DOSES TAPER DOSES WHEN STOPING), PSYCHOLOGICAL- ATC DOSING(DON'T WAIT TILL PAIN)  
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show PHYSICAL- REACTIVE FASHION DEPENDENCE... PSYCHOLOGICAL- ATC DOSING PROACTIVE- SHOULD HAVE SCHEDULE SET UP  
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ACETAMINOPHEN NARROW THERAPEUTIC EFFECT   show
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show CYSTEIN(MUCOMYST)  
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NON TOXIC IN GENERAL FOR TYLENOL   show
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show ANALGESIC, ANTIPYRETIC, ANTI-INFLAMMATORY- BETTER THEN TYLENOL FOR RHEUMATOID ARTHRITIS- INHIBITS PROSTAGLANDIN SYNTHESIS  
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show SHORT TERM-GI ULCERATION... LONG TERM- RENAL DAMAGE (TAKES DECADES)  
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show ON MORE THEN ONE DRUG THEN IS NEEDS-LASIX FROM ONE MD AND FURESOMIDE FROM OTHER MD  
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IBUPROFEN   show
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show LONG ACTING AND LONG ONSET GOOD FOR KEEPING PAIN AWAY  
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200MG IBUPROFEN PO QMORNING AND 275MG NAPROXEN PO Q12H   show
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show SEDATIVE GOAL IS CALM...HYPNOTIC GOAL IS SLEEP-CAN BE USED FOR 2 THINGS (SLEEP/CALM)  
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BENZODIAZEPINES-HYPNOTIC LOTTA   show
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ATIVAN,SERAX, RESTORIL   show
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show LONGER HALF LIFE W/ AGE SO SHOULD BE AVOIDED IN ELDERLY  
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show SO WILL HAVE HANGOVER EX VALIUM, AMBIEN  
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show SUPRESS NEURONAL FIRING-WIDE THERAPEUTIC INDEX TILL YOU ADD ETOH B/C ETOH CAN AMPLIFY 2X-200X THE EFFECT S/E SOME HAVE MILD ANTICHOLINERGIC EFFECTS, OTHERS ANTEROGRADE AMNESIA (CAN'T REMEMBER WHATS HAPPENS WHILE ON DRUG) DON'T TEACH PT WHILE USING THESE  
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ANTIPSYCHOTICS   show
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ANTIDEPRESSANTS   show
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GENERAL S/E FOR ANTIPSYCHOTICS   show
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EX HALDOL S/E   show
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ALL ANTIPSYCHOTICS ANTIDEPRESSANTS   show
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show 3 WEEKS TO 3 MONTHS (FOR MORE ORDERED THOUGHT OR RAISED MOOD)  
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show PK  
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THERAPEUTIC INDEX   show
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B-BLOCKERS W/ DIABETES   show
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PHARMACEUTICS   show
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show GIVE ALBUTEROL  
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CARDIOVASCULAR-HTN 3 PARTS KIDNEYS HEART VESSELS   show
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show ^HR AND STRENGTH (FAST) AND CONSTRICTION OF VESSLES(FAST)  
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show VESSLES CONSTRICT(FAST) KIDNEYS RETAIN FLUID(SLOW)  
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show ^HR AND STRENGTH(FAST) AND KIDNEYS FLUID RETENTION(SLOW)  
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show -PRIL. CAPTOPRIL/CAPOTEN  
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ARB's   show
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B-BLOCKERS   show
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show VERAPAMIL/CALAN DIALTIAZEM/CARDIZEM  
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ALPHA BLOCKERS   show
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show -DIPINE..DIFEDIPINE/PROCARDIA  
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FINALLY THE END- GOOD LUCK:)   show
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