| Term | Definition |
| Albuterol Drug Class | Beta-2 agonist |
| Albuterol Mechanism of Action | Stimulation of SNS beta-2 receptors
Smooth muscle relaxation of bronchioles |
| Albuterol Adverse Effects | Tachycardia, palpitations, restlessness
H/A |
| Albuterol Contraindications | Cardiac disease, hyperthyroidism |
| Albuterol Interactions | Beta blockers |
| Albuterol Nursing Indications | Monitor HR, respiratory status
Teach regarding rescue inhaler use
Use 30-60 minutes before exercise
Avoid caffeine |
| Ipratropium Drug Class | Anticholinergic |
| Ipratropium Mechanism of Action | Increased PNS stimulation on CN X
Antagonizes muscarinic receptors |
| Ipratropium Adverse Effects | Dry mouth, blurry vision, tachycardia, urinary retention, constipation |
| Ipratropium Contraindications | Narrow angle glaucoma
Bladder neck obstruction/BPH
Allergy to soy or peanuts (propellant sensitivity) |
| Ipratropium Interactions | Other anticholinergics |
| Ipratropium Nursing Indications | Monitor VS, respiratory status
Monitor UOP
Teach to void prior to drug administration
Lozenges
Fiber/fluids |
| Budesonide Drug Class | Corticosteroid |
| Budesonide Mechanism of Action | Inhibition of inflammatory response |
| Budesonide Adverse Effects | Sore throat
Xerostomia
Oral candidiasis |
| Budesonide Contraindications | Active infections
Oral lesions increase systemic absorption |
| Budesonide Nursing Indications | Monitor respiratory status, oral mucosa
Taper the dose
Rinse mouth after inhalation |
| Drug of choice for rescue inhaler | SABA - albuterol |
| Theophylline Drug Class | Methylxanthines |
| Theophylline Mechanism of Action | Smooth muscle relaxation via mobilization of calcium and activation of prostaglandins
Inhibition histamine |
| Theophylline Adverse Effects | Typically only associated with toxicity
20-25 mcg/mL: N/V/D, insomnia, diaphoresis, H/A and irritability
>30-35 mcg/mL: hyperglycemia, hypokalemia, hypotension, dysrhythmias, tachycardia, seizures, brain damage and death |
| Theophylline Interactions | Multiple interactions – including caffeine
Smoking increases metabolism of theophylline
With smoking cessation – toxicity! |
| Theophylline Contraindications | Caution with cardiac disease, hyperthyroidism |
| Theophylline Nursing Indications | Monitor VS, lung sounds
Serum drug level
Decrease caffeine intake
Toxicity treatment
Activated charcoal, lidocaine, benzodiazepines |
| Montelukast Drug Class | Leukotriene receptor antagonist |
| Montelukast Mechanism of Action | Decreases: neutrophil, eosinophil migration, aggregation, leukocyte adhesion, capillary permeability, smooth muscle contraction |
| Montelukast Adverse Effects | H/A, dizziness
Elevated LFTs
Suicidal ideation |
| Montelukast Interactions | Increases toxicity of theophylline, warfarin |
| Montelukast Nursing Indications | Monitor respiratory status
Take on empty stomach
Taper dose
Avoid triggers |