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MCPHS Therapeutics
MCPHS HIV Interactions Stuff
Drug | CYP Action |
---|---|
Theophylline | 1A2 substrate |
Haloperidol | 1A2 substrate |
Ciprofloxacin | 1A2 inhibitor |
Clarithromycin | 1A2 inhibitor, 3A4 inhibitor |
Statins | some 3A4 substrates |
Amiodarone | 3A4 substrate |
Ritonavir | 1A2 inducer, 2C9 inhibitor, 2D6 inhibitor, 3A4 substrate, 3A4 inhibitor, 3A4 inducer |
Cigarette Smoke | 1A2 inducer |
Phenytoin | 1A2 inducer, 2C9 substrate, 2C9 inducer, 2D6 inducer, 3A4 inducer |
Phenobarb | 1A2 inducer, 2C9 inducer, 2D6 inducer, 3A4 inducer |
Carbamazepine | 1A2 inducer, 2C9 inducer, 2D6 inducer, 3A4 inducer |
Warfarin | 2C9 substrate, 3A4 substrate |
Voriconazole | 2C9 substrate |
Efavirenz | 2C9 inhibitor, 3A4 substrate, 3A4 inducer |
Rifampin | 2C9 inducer, 2D6 inducer, 3A4 inducer |
Codeine | 2D6 substrate |
Methadone | 2D6 substrate |
SSRIs | 2D6 substrate, 2D6 inhibitor |
PIs | 3A4 substrate, 3A4 inhibitors |
NNRTIs | 3A4 substrate |
Benzos | 3A4 substrate |
Sildenafil | 3A4 substrate |
Vardenafil | 3A4 substrate |
Tadalafil | 3A4 substrate |
Delveradine | 3A4 substrate, 3A4 inhibitor |
Azoles | 3A4 inhibitor |
Erythromycin | 3A4 inhibitor |
Nevirapine | 3A4 substrate, 3A4 inducer |
St. Johns Wort | 3A4 inducer |
Garlic | CYP inhibitor |
Grapefruit Juice | 3A4 inhibitor |
Tramadol | 2D6 substrate |
TCA | 2D6 substrate |