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MCPHS Therapeutics
MCPHS HIV Interactions Stuff
| Drug | CYP Action |
|---|---|
| Theophylline | 1A2 substrate |
| Haloperidol | 1A2 substrate |
| Ciprofloxacin | 1A2 inhibitor |
| Clarithromycin | 1A2 inhibitor, 3A4 inhibitor |
| Statins | some 3A4 substrates |
| Amiodarone | 3A4 substrate |
| Ritonavir | 1A2 inducer, 2C9 inhibitor, 2D6 inhibitor, 3A4 substrate, 3A4 inhibitor, 3A4 inducer |
| Cigarette Smoke | 1A2 inducer |
| Phenytoin | 1A2 inducer, 2C9 substrate, 2C9 inducer, 2D6 inducer, 3A4 inducer |
| Phenobarb | 1A2 inducer, 2C9 inducer, 2D6 inducer, 3A4 inducer |
| Carbamazepine | 1A2 inducer, 2C9 inducer, 2D6 inducer, 3A4 inducer |
| Warfarin | 2C9 substrate, 3A4 substrate |
| Voriconazole | 2C9 substrate |
| Efavirenz | 2C9 inhibitor, 3A4 substrate, 3A4 inducer |
| Rifampin | 2C9 inducer, 2D6 inducer, 3A4 inducer |
| Codeine | 2D6 substrate |
| Methadone | 2D6 substrate |
| SSRIs | 2D6 substrate, 2D6 inhibitor |
| PIs | 3A4 substrate, 3A4 inhibitors |
| NNRTIs | 3A4 substrate |
| Benzos | 3A4 substrate |
| Sildenafil | 3A4 substrate |
| Vardenafil | 3A4 substrate |
| Tadalafil | 3A4 substrate |
| Delveradine | 3A4 substrate, 3A4 inhibitor |
| Azoles | 3A4 inhibitor |
| Erythromycin | 3A4 inhibitor |
| Nevirapine | 3A4 substrate, 3A4 inducer |
| St. Johns Wort | 3A4 inducer |
| Garlic | CYP inhibitor |
| Grapefruit Juice | 3A4 inhibitor |
| Tramadol | 2D6 substrate |
| TCA | 2D6 substrate |