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Phar-Hague 4
Antihypertensives
| Question | Answer |
|---|---|
| Beta blockers | Propanalol Metopralol Carvedilol |
| Propanalol MOA & admin | Nonspecific Beta blocker Oral |
| Propanalol use / side effect | Use -CHF -HTN -Angina Side effect -Hypotension -Nausea |
| Metoprolol MOA & admin | Cardioselective B1 blocker |
| Metoprolol use / side effect | Use -CHF -HTN -Angina Side effect -Hypotension -Nausea |
| Carvedilol MOA & admin | Inhibit beta/alpha adrenergic receptors Oral |
| Carvedilol use / side effect | Use -CHF Side effects -Hypotension -Nausea |
| ACE inhibitors | Captopril Ramipril |
| Captopril MOA & admin | Inhibit angiotensin converting enzyme Oral |
| Captopril use / side effect | Use -CHF -HTN -Angina Side effect -Hypotension -Cough |
| Ramapril MOA & admin | Inhibit angiotensin converting enzyme Oral |
| Ramapril use / side effect | Use -CHF -HTN -Angina Side effect -Hypotension -Cough |
| Angiotensin receptor blockers | Losartan Valsartan |
| Losartan MOA & admin | Inhibit AT-II 1 receptors Oral |
| Losartan use / side effect | Use -CHF -HTN -Angina Side effect -Hypotension -No cough |
| Valsartan MOA & admin | Inhibit AT-II 1 receptors Oral |
| Valsartan use / side effect | Use -CHF -HTN -Angina Side effect -Hypotension -No cough |
| Aliskiren MOA & admin | -Renin inhibitor -Oral |
| Aliskiren use / side effect | Use -CHF -HTN -Angina Side effect -Hypotension -No cough |
| Bosentan MOA & admin | -Endothelin receptor inhibitor -Oral |
| Bosentan use / side effect | Use -Pulmonary hypertension Side effect -Headache |
| Hydralazine MOA & admin | -Vasodilator -K+ channel opener -Oral |
| Hydralazine use / side effect | Use -Hypertension Side effect -Hypotension -Tachycardia |
| Diuretics | Hydrochlorothiazide Furosemide |
| Hydochlorothiazide MOA & admin | Inhibit Na/Cl co-transporter, DT Oral |
| Hydochlorothiazide use / side effect | Use -CHF -Hypertension -Edema Side effects -Hyponatremia |
| Furosemide MOA & admin (Lasix) | Loop diuretic, inhibit Na/K/2Cl transpoter Oral |
| Furosemide use / side effect | Use -CHF -Hypertension -Edema Side effect -Hypokalemia |
| Ca2+ channel blockers | Verapamil Diltiazem Nifedipine |
| Verapamil MOA & admin | Voltage gated Ca channel nhibitor, cardiac Oral |
| Verapamil use / side effect | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |
| Diltiazem MOA & admin | Voltage gated Ca channel nhibitor, cardiac Oral |
| Diltiazem use / side effect | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |
| Nifedipine MOA & admin | Voltage gated Ca channel inhibitor, SMOOTH MUSCLE Oral |
| Nifedipine use / side effect | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |
| Prazosin MOA & admin | Alpha 1 blocker Oral |
| Prazosin use / side effect | Use -BPH -HTN Side effects -Orthostatic hypotension |
| Clonidine MOA & admin | Alpha 2 agonist Oral |
| Clonidine use / side effect | Use -HTN -ADHD Side effects -Dry mouth -Fatigue |