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Phar - Hague 3
Angina, Vasodilators, CHF
| Question | Answer |
|---|---|
| Beta-blockers | Propanolol Atenolol |
| Propranolol properties | non selective beta-adrenergic receptor antagonist Oral |
| Propanolol use / side effects | Use -CHF -Hypertension -Angina Side effects -Nausea -Hypotension |
| Atenolol properties | selective beta1-adrenergic receptor antagonist Oral |
| Atenolol use / side effects | Use -CHF -Hypertension -Angina Side effects -Nausea -Hypotension |
| Vasodilators | Nitroglycerine Isosorbide dinitrate |
| Nitroglycerine properties | Donate NO, increase cGMP in SMC, PKG activity, vasodilation Oral |
| Nitroglycerine use / side effects | Use -Acute decompensated HF -Angina Side effects -Hypotension -Tachycardia |
| Isosorbide dinitrate properties | Donate NO, increase cGMP in SMC, PKG activity, vasodilation Oral |
| Isosorbide dinitrate use / side effects | Use -Acute decompensated HF -Angina Side effects -Hypotension -Tachycardia |
| PDE Inhibitors | Sildenafil |
| Sildenafil properties | Inhibitor of cGMP phosphodiesterase Oral |
| Sildenafil use / side effects | Use -ED -BPH -Pulmonary hypertension Side effects -Hypotension -Vision |
| Ca2+ channel antagonists | Verapamil Diltiazem Nifedipine |
| Verapamil properties | Voltage gated Ca channel inhibitor, cardiac/VSM Oral |
| Verapamil use / side effects | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |
| Diltiazem properties | Voltage gated Ca channel inhibitor, cardiac/VSM Oral |
| Diltiazem use / side effects | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |
| Nifedipine properties | Voltage gated Ca channel inhibitor, VSM only Oral |
| Nifedipine use / side effects | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |