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NAPLEX2
| Question | Answer | |
|---|---|---|
| Duragesic | Fentanyl | Mu AgonistTransdermal |
| Actiq | Fentanyl | Mu AgonistLozenge |
| Fentora | Fentanyl | Mu AgonistODT |
| Dilaudid | Hydromorphone | Mu AgonistTablet/Liquid/Injection |
| Levo-Dimoran | Levorphanol | Mu AgonistTab/Inj |
| Demerol | Meperidine | Mu AgonistObstetric use/Metabolite=seizures |
| Dolophine | Methadone | Mu AgonistTdP |
| Methadose | Methadone | Mu AgonistTdP |
| Roxanol | Morphine | Mu AgonistImmediate Release |
| Duramorph | Morphine | Mu Agonist |
| Astramorph | Morphine | Mu Agonist |
| Avinza | Morphine | Mu AgonistControlled Release Tab |
| Kadian | Morphine | Mu AgonistControlled Release |
| MS Contin | Morphine | Mu AgonistControlled Release |
| Oramorph | Morphine | Mu AgonistControlled Release |
| Roxicodone | Oxycodone | Mu AgonistMild pain |
| OxyIR | Oxycodone | Mu AgonistImmediate release/mild pain |
| RoxiCodone | Oxycodone | Mu Agonistmild pain |
| Magnacet | Oxycodone+APAP | Mu Agonistmild pain |
| Roxicet | Oxycodone+APAP | Mu AgonistMild Pain |
| Tylox | Oxycodone+APAP | Mu AgonistMild pain |
| OxyContin | Oxycodone | Mu Agonistmild painControlled release |
| Oxymorphone | Oxymorphone | Mu Agonist |
| Opana | Oxymorphone | Mu Agonistimmediate release |
| Opana ER | Oxymorphone | Mu agonistcontrolled release |
| Reprexin/Vicodin/Lortab/Hycet/Zydone/Vicoprofin | HydroconeAPAP or IBU | mild-moderate pain |
| DarvcetNDarvon | Propoxyphene | Mild-moderate painwk analgesic and increased ADR |
| Talwin | Pentazocine | Agonist/AntagonistPartial AgonistDetox |
| Talwin NS | Pentazocine+Naloxone | Agonist/AntagonistPartial AgonistDetox |
| Talwin Compound | Pentazocine+ASA | Agonist/AntagonistPartial AgonistDetox |
| Stadol | Butorphanol | Agonist/AntagonistPartial AgonistDetox Injection/Nasal |
| Nalbuphine | Agonist/AntagonistPartial AgonistDetox Injection | |
| Buprenex | Buprenorphine | Agonist/AntagonistPartial AgonistDetox Injection |
| Narcan | Naloxone | Opioid antagonist |
| Revia | Naltrexone | Opioid antagonisttabletEtOH |
| Vivitrol | Naltrexone | Opioid antagonistinjectionEtOH |
| Voltaren | Diclofenac | NSAID |
| Cataflem | Diclofenac | NSAID |
| Lodine | Etodolac | NSAIDLow GI risk |
| Indocin | Indomethacin | NSAIDHigh GI risk |
| Relafen | Nabumetone | NSAIDLow GI risk |
| Tolectin | Tolmetin | NSAID |
| Clinorial | Sulindac | NSAID |
| Meclomen | Meclofenamate | NSAID |
| Feldene | Piroxicam | NSAIDHigh GI risk |
| Nalfon | Fenoprofen | NSAID |
| Ansaid | Flurbiprofen | NSAID |
| MotrinAdvil | IBU | NSAID |
| OridisOruvil | Ketoprofen | NSAID |
| NaprosynAleve | Naproxen | NSAID>12 yo |
| Daypro | Oxaprozin | NSAID |
| Celbrex | Celexocib | Cox2 inhibitor |
| Toradol | Ketorlac | NSAID |
| Dolobid | Diflunisal | NSAID |
| Mobic | Meloxicam | NSAIDLow GI risk |
| Ponstel | Mefenamic Acid | NSAID |
| Diuril | Chlorothiazide | Thiazide DiureticIncrease BG, Decrease K, sun sensitive |
| Hygroton | Chlorthiazidone | Thiazide DiureticIncrease BG, Decrease K, sun sensitive |
| Hylidone | Chlorthiazidone | Thiazide DiureticIncrease BG, Decrease K, sun sensitive |
| HydroDiuril | HCTZ | Thiazide DiureticIncrease BG, Decrease K, sun sensitive |
| Mykrox | Metolazone | Thiazide DiureticIncrease BG, Decrease K, sun sensitiveEffective when GFR<30 |
| Zaroxolyn | Metolazone | Thiazide DiureticIncrease BG, Decrease K, sun sensitive Effective when GFR<30 |
| Lozol | Indapamide | Thiazide DiureticIncrease BG, Decrease K, sun sensitive |
| OsmitrolResectisol | Manitol | Osmotic diuretic Increase K, pulmonary edema |
| Bumex | Bumetanide | Loop diureticIncrease BG, Decrease K, ototoxicity, use for Class C HF; sulfa |
| Lasix | Furosemide | Loop diureticIncrease BG, Decrease K, ototoxicity, use for Class C HF; sulfa |
| Demadex | Torsemide | Loop diureticIncrease BG, Decrease K, ototoxicity, use for Class C HF; sulfa |
| Edecrin | Ethacrynic acid | Loop diureticIncrease BG, Decrease K, ototoxicity, use for Class C HF |
| Midamore | Amiloride | K+ SparingIncrease K, Increase BG, sexual dysfunction |
| Dyrenium | Triamterene | K+ SparingIncrease K, Increase BG, sexual dysfunction |
| Aldactone | Spironolactone | Aldosterone Receptor Blocker OR Aldosterone AntagonistHF/LVEF, increase K, gnecomastic, irregular menses |
| Inspra | Eplerone | Aldosterone Receptor Blocker OR Aldosterone AntagonistHF/LVEF, increase K, gnecomastic, irregular menses |
| Hylorel | Guanadrel | PG Adrenergic Blocker (alpha2 Ag) |
| Ismelin | Guanathidine | PG Adrenergic Blocker (alpha2 Ag) |
| Serpasil | Reserpine | PG Adrenergic Blocker (alpha2 Ag) |
| Catapress | Clonidine | Alpha2 AgonistSedation, fluid retention, sexual dysfunction, rebound HTN |
| Wytensin | Guanabenz | Alpha2 AgonistSedation, fluid retention, sexual dysfunction, rebound HTN |
| Tenex | Guafacine | Alpha2 AgonistSedation, fluid retention, sexual dysfunction, rebound HTN |
| Aldomet | Methyldopa | Alpha2 AgonistSedation, fluid retention, sexual dysfunction, rebound HTN |
| Cardura | Doxazosin | Alpha1 Blocker(VD)QHS, priapsm, peripheral edema |
| Minipress | Prazosin | Alpha1 Blocker(VD)QHS, priapsm, peripheral edema |
| Hytrin | Terzosin | Alpha1 Blocker(VD)QHS, priapsm, peripheral edema |
| Tenormin | Atenolol | BBMigrain Prevention, Cardio,rebound HTN, Increase BG, sexual dysfunction |
| Zebeta | Bisoprolol | BBHF indication, Cardio,rebound HTN, Increase BG, sexual dysfunction |
| Lopressor | Metoprolol tartrate | BBMigrain Prevention, Cardio,rebound HTN, Increase BG, sexual dysfunction |
| Toprol XL | Metoprolol succinate | BBMigrain Prevention, Cardio,rebound HTN, Increase BG, sexual dysfunction, HF indication |
| Corgard | Nadolol | BBrebound HTN, Increase BG, sexual dysfunction |
| Inderal | Propranolol | BBMigrain Prevention, sedation,rebound HTN, Increase BG, sexual dysfunction |
| Blocadren | Timolol | BBMigrain Prevention, rebound HTN, Increase BG, sexual dysfunction |
| Coreg | Carvidilol | BBHF indication, rebound HTN, Increase BG, sexual dysfunction |
| NormodyneTrandate | Labetolol | rebound HTN, Increase BG, sexual dysfunction |
| Apresoline | Hydralazine | Direct VDTachycardia, fluid retention |
| Loniten | Minoxidil | Direct VDTachycardia, fluid retention, hirsutism |
| Cardizem, Dilacar, Tiazac | Diltiazem | Non-CCB (- inotrope)-Gingival hyperplasia, edema |
| Calan, Isoptan, Covera HS, Valeran PM | Verapamil | Non-CCB (- inotrope)-Gingival hyperplasia, edema |
| Norvasc | Amlodipine | Di-CCBGingival hyperplasia, edema |
| Plendil | Felodipine | Di-CCBGingival hyperplasia, edema |
| Dynacirc | Isradipine | Di-CCBGingival hyperplasia, edema |
| Cardene | Nicardipine | Di-CCBGingival hyperplasia, edema |
| Procardia, Adalat | Nifedipine | Di-CCBGingival hyperplasia, edema |
| Lotensin | Benazepril | ACEI-angioedema, category X, increase K, cough |
| Capoten | Captropil | ACEI-angioedema, category X, increase K, cough |
| Vasote | Enalapril | ACEI-angioedema, category X, increase K, cough |
| Monopril | Fosinopril | ACEI-angioedema, category X, increase K, cough |
| Univasc | Moexipril | ACEI-angioedema, category X, increase K, cough |
| Accupri | Quinapril | ACEI-angioedema, category X, increase K, cough |
| Altace | Rampipril | ACEI-angioedema, category X, increase K, cough |
| Mavik | Tranodopril | ACEI-angioedema, increase K, cough, category X |
| Prinivil, Zestril | Lisinopril | ACEI-angioedema, category X, increase K, cough |
| Atacand | Cardesartan | ARB-angioedema, increase K, category X, HF indication |
| Tevetan | Eprosartan | ARB-angioedema, increase K, category X |
| Avapro | Irbesartan | ARB-angioedema, increase K, category X |
| Cozaar | Losartan | ARB-angioedema, increase K, category X |
| Micardis | Telmesartan | ARB-angioedema, increase K, category X |
| Diovan | Valsartan | ARB-angioedema, increase K, category X, HF indication |
| Benicar | Olmesartan | ARB-angioedema, increase K, category x |
| Tekturna | Aliskiren | Direct Renin Inhibitor-angioedema, increase K, category X, D |
| AntiHTN Migraine Px | Timolol, propranolol, atenolol | - |
| AntiHTN HF indication | Diovan, Atacand, Metoprolol, carvidiol, bisoprolol | - |
| AntiHTN Decrease K | Thiazide diuretic, Loop diuretic | - |
| AntiHTN Increase K | K+ Sparing, ACEI, ARB, Direct Renin, Osmotic diuretic, Aldosterone Ant | - |
| AntiHTN angioedema | ACEI, ARB, Direct Renin Inhibitor | - |
| AntiHTN edema | CCB, Direct VD, alpha1 blocker, alpha2 agonist | - |
| AntiHTN sedation | alpha2 agonist, propranolol | - |
| AntiHTN gingival hyperplasia | CCB | - |
| AntiHTN priapsim | alpha1 blocker | - |
| AntiHTN rebound HTN | alpha2 agonist, BB- | |
| Class I Antiarrythmic | Quinidine, procainamide, disopyramide, morcinzine, lidocaine, tocainide, mexiletine, flecainide, propafenone | Ear/eye=Qunidine; -inotrope/ anticholinergic = disopyramide; seizures + CNS toxicity = lidocaine; metallic taste = propafenone ; increase mortality in HF; negative inotrope; TdP |
| Class II Antiarrythmic | BB-Metoprolol, Propranolol, Esmolol | RATE control; rebound HTN; Caution HF, Asthma, DM |
| Class III Antiarrythmic | Amiodarone (Cordarone/Pacerone), Sotolol (Betapace), Ibutiloide (Covert), Dofetilide (Tikosyn) | RHYTHM, TdP; amiodarone = visual, liver, cardiac, pulmonary, photo |
| Class IV Antiarrythmic | Verapamil & Diltiazem | RATE, negative inotrope t/f avoid in HF |
| Atopen | Atropine | Anticholinergic to increase CO, dry secretions, 5HT ant |
| Adenocard | Adenosine | Slows conduction (VD) |
| Epinephrine | Relax Smooth muscle | |
| Lanoxin, Lanoxicaps | Digoxin | + inotrope; CV, GI, neurological, DI, TDM (>2=tox), renal |
| Vasodilators | Nitropursside (Nipride), Nitroglycerin (Nitro-Bid, Nitrostat), Nesiritide (Natrecor) | Hypotension and HA, nitroprusside tox (cyanide), nesiritide increases diuresis and tachycardia; NTG tachycardia and tolerance |
| Intotropes | Dopamine (Intropin), Dobutamine (Dobutrex), Milrinone (Primacor) | Dobutamine for hypotensive pts, adjust milrinone for renal insufficiency |
| Antiarrythmic - inotrope | Class I, Class IV | - |
| Antiarrythmic + inotrope | Digoxin, Dobutamine, Dopamine, milrinone | - |
| Antiarrythmic CI HF | Class I, Class II, Class IV | - |
| Antiarrythmic TdP | Class I, Class III | - |
| Antiarrythmic eye | Qunidine, amiodarone, dig | - |
| Antiarrythmic ear | qunidine | - |
| Antiarrythmic liver | amiodarone | - |
| Antiarrythmic kidney | dig and milrinone | - |
| Antiarrythmic photosensitive | amiodarone | - |
| Ranexa | Ranolazine | Management of chronic stable angina |
| Plavix | Clopidogrel | Antiplatelet, increase bleed |
| Ticlid | Ticlopidine | Antiplatelet, increase bleed, thrombocytopenia, neutropenia, liver |
| ReoPro | Abciximab | Antiplatelet (GLY IIb/IIIa), thrombocytopenia, renal, long DOA, PCI, allergy |
| Integrilin | Eptifibate | Antiplatelet (GLY IIb/IIIa), thrombocytopenia |
| Aggrastat | Tirofiban | Antiplatelet (GLY IIb/IIIa), thrombocytopenia |
| Aggrenox | ASA + Dipyridamole | Antiplatelet |
| Lovenox | Enoxaparin | LMWH, Factor Xa, Bleed, thrombocytopenia, epidural/spinal anetheisa warning, renally eliminated |
| Fragmin | Dalteparin | LMWH, Factor Xa, Bleed, thrombocytopenia, epidural/spinal anetheisa warning |
| Arixtra | Fondaparinux | Factor Xa Inhibitor, bleed, thrombocytopenia |
| Angiomax | Bivalirudien | Direct Thrombin Inhibitor |
| Argatroban | DTI | |
| Iprivask | Desirudin | DTI |
| Refludan | lepirudin | DTI |
| Protamine | - | - |
| Coumadin | Warfarin | Anticoagulant... |
| Streptase | Streptokinase | Thrombolytic |
| Alteplase | tPA tissue plasminogen activator | thrombolytic |
| Retevase | Reteplase | Thrombolytic |
| TNKase | Tenectase | Thrombolytic |
| Bleed | warfarin, ASA, clopidogrel, Ticlid, Abc/tiro/ept, thrombolytics, hep, LMWH, fondaparinux | - |
| Thrombocytopenia | LMWH, Fondaparinux, Hep, Ticlid, Abc/ept/tiro | Use DTI |
| Renal | Enoxaprin, ABC, ASA | - |
| Liver | Ticlid | - |
| Paroxysmal supraventricular Tachycardia | Adenosine | - |
| Sinus bradycardis | Atropine | - |
| AV Block | Atropine | - |
| Atrial Fibrillation | Rhythm (young/ hemodynamically unstable/ no HF)=Class III AADRate+Warfarin (stroke, embolism, TIA< >75, HTN, DM, LF, HF)=Class II Or IV or Dig | No P Wave |
| Premature Ventricualar Contraction (PVC) | If HF=BBDofetilide (Tikosyn) | - |
| Ventricular Fibrillation | Life Support, Epi, Vasopressor | Scarry teeth, sudden cardiac death |
| Ventricular Tachycardia | CPR, Epi, Vasopressor | Wide QRS |
| Torsades de Pointes | Mg, K | Twist QRS |
| Stable Angina Treatment | Treat if greater than 1 episode per day=BB, CCB, LA nitrate, Ranexa, AntiPLT, ACEI, lipid; NTG for acute attach | - |
| Unstable Angina Treatment | Invasive=MONA+AntiCOAG+Plavix+Abc; Conservative=MONA+AntiCOAG(LMWH/UFH)+Plavix+EPT/TIRO | - |
| STEMI | MONA+Reperfusion(CABG /PCI <90min /Thrombolytics <30 min) + AntiCOAG | Discharge=BB+ACEI+Statin+SC +NTG+ASA |
| ID Quality Indicators for MI | ASA @ arrival, BB @ arrival, Thrombolytic (30) for STEMI, PCI (90), ASA @ DC, BB @ DC, ACEI/ARB for LVD, Smoking cessation | - |
| AntiPLT duration of therapy | ASA 81 mg indefinantly; 325 PCI X1 month BMS, X3 month SES, X6 month PES | Clopidogrel LD 300-600mg then 75mg daily X |
| Lower LDL | Statin, Niacin, Resin, Omega3FA | - |
| Increase HDL | Niacin, Fibrinic Acid | - |
| Lower TG | Niacin, Fibrinic Acid, Omega3FA | - |
| LFT | Statin, Niacin, Fibrinic Acid, Cholesterol Inhibitor | - |
| Glucose | Niacin | - |
| Uric acid | Niacin | - |
| CI>TG | BAS | - |
| Myopathy | Statin, Niaci, Fibrinic Acid | - |
| Sublimaze | Fentanyl | Mu AgonistInjection |