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B Pharmaco Ex2
PCOL Cholinergic Drug/Extra Key Info
| Drug | Extra/ Key Info |
|---|---|
| Acetylcholine Methacholine Carbachol Bethanechol | --- |
| Pilocarpine Cevimeline | Treatment for Dry Mouth (enhance salivation) Treatment of Glaucoma |
| Atropine | Treatment for Organophosphate Poisoning (severe DUMBBELSS) Treatment for Muscurinic Agonist OD |
| Scopolamine | Motion Sickness |
| Benztropine (Cogentin) | Treat Parkinson's |
| Tropicamide | Pupil Dilation (M3) |
| Ipratropium (Atorvent) | Short-acting muscurinic antagonist (SAMA) |
| Tiotropium (Spiriva) | Long-acting muscurinic antagonist (LAMA) |
| Aclidinium Umeclidinium | Long-acting muscurinic antagonist (LAMA) |
| Oxybutynin (diTROPan) Tolterodine Fesoterodine Solifenacin Darifenacin Trospium | Solifenacin, Darifenacin and Trospium are Most Selective for M3-->least likely to cause DUMBbELSS Treats Overreactive Bladder |
| Nitroglycerine Nitroprusside Isosobide di/monitrate | cGMP is a Potent Vasodilator |
| Sildenafil (Viagra) Tadalafil (Cialis) Vardenafil | Blocks enzyme that breaks down cGMP=more cGMP Used to treat Erectile Dysfunction |