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B Pharmaco Ex2
PCOL Adrenergic Drugs/MOA
Drug | MOA |
---|---|
Phenylephrine | a1 agonist |
Cocaine | NE Reuptake Inhibitor |
Dextroamphetamine/Amphetamine (Addy) Methylphenidate (Concerta, Ritalin) Lisdexamphetamine (Vyvanse) Dexmethylphenidate (Focalin) | Stimulate Pre-Synaptic release of NE & DA |
Phenelzine | Non-Selective MOA-A & MOA-B Irreversible Antagonist |
Selegiline Rasagiline | Selective MAO-B Irreversible Antagonist |
Prazosin Terazosin (Hytrin) Doxazosin (Cardura) Tamsulosin (Flomax) -> alpha1a | Selective a1 Reversible Antagonist |
Phenoxybenzamine | Non-Selective a1 & a2 Irreversible Antagonist *Decreases Peripheral Resistance |
Mirtazapine (Remeron) | Non-Selective a1/a2 antagonist, Muscurinic Antagonists, H1 Antagonist, 5-HT 2a Antagonist |
Clonidine (Catapres) Brimonidine (Alphagan P) Tizanidine (Zanaflex) Guanfacine (Intuniv) Dexmedetomidine (Precedex) | a2 agonist |