click below
click below
Normal Size Small Size show me how
B Pharmaco Ex2
PCOL Cholinergic Drug/MOA
| Drug | MOA |
|---|---|
| Methacholine Carbachol Bethanechol | Non-Selective Muscurinic Agonist (M1, M2, M3) *Agonist |
| Pilocarpine Cevimeline | Non-Selective Muscurinic Agonist (M1, M2, M3) *Agonist |
| Atropine | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
| Scopalamine | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
| Benztropine (Cogentin ) | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
| Tropicamide | Muscurinic Antagonist |
| Ipratropium (Atorvent) | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
| Tiotropium (Spiriva) | SELECTIVE Muscurinic Antagonist (M1 & M3) |
| Aclidinium Umeclidinium | Muscurinic Antagonist |
| Oxybutynin (diTROPan) Tolterodine Fesoterodine Solifenacin Darifenacin Trospium | Non-Selective Muscurinic Antagonist (M1, M2, M3) *All more selective for M3* |
| Nitroglycerine Nitroprusside Isosobide di/monitrate | Donate nitric oxide NO-->sGC-->INCREASE cGMP |
| Sildenafil (Viagra) Tadalafil (Cialis) Vardenafil | Blocks PDE-->INCREASE cGMP |