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B Pharmaco Ex2
PCOL Cholinergic Drug/MOA
Drug | MOA |
---|---|
Methacholine Carbachol Bethanechol | Non-Selective Muscurinic Agonist (M1, M2, M3) *Agonist |
Pilocarpine Cevimeline | Non-Selective Muscurinic Agonist (M1, M2, M3) *Agonist |
Atropine | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
Scopalamine | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
Benztropine (Cogentin ) | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
Tropicamide | Muscurinic Antagonist |
Ipratropium (Atorvent) | Non-Selective Muscurinic Antagonist (M1, M2, M3) *Antagonist *Anti-cholinergic |
Tiotropium (Spiriva) | SELECTIVE Muscurinic Antagonist (M1 & M3) |
Aclidinium Umeclidinium | Muscurinic Antagonist |
Oxybutynin (diTROPan) Tolterodine Fesoterodine Solifenacin Darifenacin Trospium | Non-Selective Muscurinic Antagonist (M1, M2, M3) *All more selective for M3* |
Nitroglycerine Nitroprusside Isosobide di/monitrate | Donate nitric oxide NO-->sGC-->INCREASE cGMP |
Sildenafil (Viagra) Tadalafil (Cialis) Vardenafil | Blocks PDE-->INCREASE cGMP |