click below
click below
Normal Size Small Size show me how
B Pharmaco Ex2
PCOL Neuromuscular Drug/MOA
Drug | MOA |
---|---|
Acetylcholine | Depolarizing agent (Nicotinic & Muscurinic) *Agonist |
Varenicline (Chantix) | a4/B2 Nn Partial Agonist *Agonist |
Succinylcholine | Depolarizing agent (Nm Blockade-Nicotinic) *Agonist |
Physostigmine | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
Donepezil Rivastigmine Galantamine | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
PyriDOstigmine Neostigmine | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
Edrophonium | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
Echothiophate | Organophosphate inhibitor of Ache enzyme *Indirect Antagonist |
Botulinum | Prevent ACH release |
Mivacurium Vecuronium Rocuronium Pancuronium Tubocuranine | NON-depolarizing agent *Direct competitive antagonist-->Binds to Ach binding space |