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B Pharmaco Ex2
PCOL Neuromuscular Drug/MOA
| Drug | MOA |
|---|---|
| Acetylcholine | Depolarizing agent (Nicotinic & Muscurinic) *Agonist |
| Varenicline (Chantix) | a4/B2 Nn Partial Agonist *Agonist |
| Succinylcholine | Depolarizing agent (Nm Blockade-Nicotinic) *Agonist |
| Physostigmine | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
| Donepezil Rivastigmine Galantamine | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
| PyriDOstigmine Neostigmine | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
| Edrophonium | Cholinesterase Inhibitor (ACHe Antagonist) *Indirect Antagonist |
| Echothiophate | Organophosphate inhibitor of Ache enzyme *Indirect Antagonist |
| Botulinum | Prevent ACH release |
| Mivacurium Vecuronium Rocuronium Pancuronium Tubocuranine | NON-depolarizing agent *Direct competitive antagonist-->Binds to Ach binding space |