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2009 Top 200 Drugs
Top 200 Prescribed Drugs of 2009...(Only 190 because I got sick of making them)
Question | Answer |
---|---|
Atenolol | Tenormin Beta Blocker (Beta 1 selective) |
Metoprolol | Lopressor (Tartrate) Toprol XL (Succinate) Beta Blocker (Beta 1 selective) Shown to decrease mortality in heart failure |
Carvedilol | Coreg, Coreg CR Beta Blocker Shown to decrease mortality in heart failure |
Labetalol | Trandate Beta blocker |
Nadolol | Corgard Beta blocker |
Propranolol | Inderal, Inderal LA, InnoPran XL Beta Blocker |
Benazepril | Lotensin ACE Inhibitor |
Captopril | Capoten ACE Inhibitor |
Enalapril | Vasotec ACE Inhibitor |
Fosinopril | Monopril ACE Inhibitor |
Lisinopril | Prinivil, Zestril ACE Inhibitor |
Quinapril | Accupril ACE Inhibitor |
Ramipril | Altace ACE Inhibitor |
Candesartan | Atacand ARB |
Irbesartan | Avapro ARB |
Losartan | Cozaar ARB |
Olmesartan | Benicar ARB |
Telmisartan | Micardis ARB |
Valsartan | Doivan ARB |
Amlodipine | Norvasc Calcium channel blocker (DHP->Selective to vasculature, more potent vasodilation, no effect on HR) |
Felodipine | Plendil Calcium channel blocker (DHP->Selective to vasculature, more potent vasodilation, no effect on HR) |
Nifedipine | Adalat CC, Afeditab CR, Nifediac CC, Nifedical XL, Procardia EL Calcium channel blocker (DHP->Selective to vasculature, more potent vasodilation, no effect on HR) |
Diltiazem | Cardizem CD, Cardizem LA, Cartia XT, Dilacor XR, Taztia XT, Tiazac Calcium channel blocker (Non-DHP->Nonselective, less peripheral vasodilation, negative chronotropes, decrease HR) |
Verapamil | Calan, Calan SR, Covera-HS, Isoptin SR, Verelan, Verelan PM (Non-DHP->Nonselective, less peripheral vasodilation, negative chronotropes, decrease HR) |
Doxazosin | Cardura Alpha-1 receptor antag |
Terazosin | Hytrin Alpha-1 receptor antag |
Clonidine | Catapres, Catapres-TTS Central alpha-2 receptor agonist |
Methyldopa Not Top 200 but good to know | Aldomet Central alpha-2 receptor agonist |
Hydralazine | Apresoline Direct vasodilator (arterial) |
Minoxidil Not top 200 but good to know | Loniten Direct vasodilator (arterial) |
Niacin | Niaspan Decreases VLDL production in liver leading to decreased synthesis of LDL |
Fenofibrate | Antara, Lipofen, Lofibra, TriCor, Triglide Fibric acid derivative (Increases activity of lipoprotein lipase which increase catabolism of VLDL which decreases triglycerides) |
Gemfibrozil | Lopid Fibric acid derivative (Increases activity of lipoprotein lipase which increase catabolism of VLDL which decreases triglycerides) Avoid with statins (myopathy) |
Omega 3 fatty acids | Lovaza |
Atorvastatin | Lipitor HMG CoA reductase inhibitor Rosuvastatin > atorvastatin > simvastatin > pravastatin = lovastatin > fluvastatin |
Fluvastatin | Lescol, Lescol XL HMG CoA reductase inhibitor Rosuvastatin > atorvastatin > simvastatin > pravastatin = lovastatin > fluvastatin |
Lovastatin | Altoprev, Mevacor HMG CoA reductase inhibitor Rosuvastatin > atorvastatin > simvastatin > pravastatin = lovastatin > fluvastatin |
Pravastatin | Pravachol HMG CoA reductase inhibitor Rosuvastatin > atorvastatin > simvastatin > pravastatin = lovastatin > fluvastatin |
Simvastatin | Zocor HMG CoA reductase inhibitor Rosuvastatin > atorvastatin > simvastatin > pravastatin = lovastatin > fluvastatin |
Rosuvastatin | Crestor HMG CoA reductase inhibitor Rosuvastatin > atorvastatin > simvastatin > pravastatin = lovastatin > fluvastatin |
Ezetimibe | Zetia Cholesterol absorption inhibitor (prevents absorption of cholesterol from small intestine) |
Bumetanide | Bumex Loop diuretic (More bioavailable than furosemide) |
Furosemide | Lasix Loop diuretic |
Torsemide | Demadex |
Digoxin | Digitek, Lanoxin Inhibits Na+/K+ ATPase pump leading to increased intracellular Ca2+ leading to increased mycardial contractility. Also causes decreased neurohormonal activation |
Spironolactone | Aldactone Nonselective aldosterone receptor antagonist (inhibits effects of aldosterone thereby decreasing remodeling and Na+/water retention) |
Amiodarone | Cordarone, Pacerone K+ channel blocker, Na+ channel blocker, CCB properties and nonselective BB properties |
Penicillin VK | Veetids Natural Penicillin |
Amoxicillin | Amoxil, Trimox Aminopenicillin |
Amoxicillin plus clavulanic acid | Augmentin Aminopenicillin |
Cephalexin | Keflex First generation cephalosporin (PO) |
Cefprozil | Cefzil 2nd generation cephalosporin (PO) |
Cefuroxime | Ceftin, Zinacef 2nd generation cephalosporin (PO) |
Cefdinir | Omnicef 3rd generation cephalosporin (PO) |
Azithromycin | Zithromax, Zmax Macrolide |
Clarithromycin | Biaxin Macrolide |
Doxycycline | Doryx, Vibramycin Tetracycline |
Minocycline | Dynacin, Minocin Tetracycline |
Ciprofloxacin | Cipro, Proquin XR Fluoroquinolone |
Levofloxacin | Levaquin Fluoroquinolone |
Sulfamethoxazole SMX and trimethoprim TMP | Bactrim, Septra Sulfonamide |
Metronidazole | Flagyl, Metrogel, Noritate, Vandazole |
Fluconazole | Diflucan Azole antifungal |
Ketoconazole | Nizoral Azole antifungal |
Nystatin | Mycostatin Antifungal |
Acyclovir | Zovirax Antiviral |
Valacyclovir | Valtrex Antiviral |
Oseltamivir | Tamiflu Antiviral |
Fluticasone | Flovent, Flovent HFA Glucocorticoid receptor agonist (corticosteroid) |
Budesonide | Pulmicort, Respules Glucocorticoid receptor agonist (corticosteroid->the only nebulized one) |
Mometasone | Asmanex Glucocorticoid receptor agonist (corticosteroid) |
Salmeterol | Serevent Long acting beta 2 agonist |
Montelukast | Singulair Leukotriene receptor antagonist |
Albuterol | Ventolin, Proventil Short acting beta 2 agonist |
Levoalbuterol | Xopenex, Xopenex HFA Short acting beta 2 agonist |
Fluticasone/Salmeterol | Advair Combo corticosteroid and long acting beta 2 agonist |
Varenicline | Chantix Partial nicotinic receptor agonist/antag |
Bupropion | Zyban 150-300mg/day Smoking cessation |
Ipratropium | Atrovent, Atrovent HFA Anticholinergic |
Tiotropium | Spiriva Anticholinergic |
Ipratropium/Albuterol | Combivent Combination of anticholinergic and short acting beta2 agonist |
Formoterol | Performist Long acting beta 2 agonist |
Insulin Aspart | NovoLog Rapid acting insulin |
Insulin Lispro | Humalog Rapid acting insulin |
NPH Neutral protamine hagedorn | Humulin N Short acting insulin |
Insulin Glargine | Lantus Long acting insulin |
75% Lispro protamine/25% lispro | Humalog 75/25 |
50% Lispro protamine/50% lispro | Humalog Mix 50/50 |
70% Insulin aspart protamine/30% aspart | NovoLog 70/30 |
70% NPH/30% regular | 70/30 |
Glyburide | Micronase Sulfonylurea |
Glipizide | Glucotrol, Glucotrol XL Sulfonylurea |
Metformin | Glucophage, Glucophage XR Biguanide |
Rosiglitazone | Avandia Thiazolidinedione |
Pioglitazone | Actos Thiazolidinedione |
Exenatide | Byetta GLP1 Inhibitor |
Sitagliptin | Januvia Dipeptidyl-peptidase 4 inhibitor |
Sitagliptin/metformin | Janumet |
Glyburide/metformin | Glucovance |
Rosiglitazone/metformin | Avandamet |
Levothyroxine | Synthroid, Levoxyl, Levothroid, Unithroid T4 |
Desiccated thyroid | Armour, Thyroid T4 80% T3 20% |
Finasteride | Proscar, Propecia alpha-5 reductase inhibitor |
Carbamazepine | Tegretol Inhibits voltage-gated sodium ion channels |
Valproic acid | Depakote, Depakote ER, Depakene, Depacon Increases GABA |
Phenytoin | Dilantin Promotes sodium efflux |
Oxcarbazepine | Trileptal Inhibits voltage-gated sodium ion channels |
Gabapentin | Neurontin similar to GABA NO DRUG INTERACTIONS |
Lamotrigine | Lamictal Inhibits voltage-gated sodium ion channels |
Topiramate | Topamax Inhibits voltage-gated sodium ion channels, augments GABA activity |
Levetiracetam | Keppra |
Phenobarbital | Solfoton |
Selegiline Not Top 200 but good to know | Eldepryl, emsam, Zelapar MAOB inhibitor, inhibits levodopa breakdown |
Carbidopa/levodopa | Sinemet, Sinemet CR, Parcopa |
Parmipexole | Mirapex Dopamine agonist |
Ropinirole | Requip Dopamine agonist |
Benztropine | Cogentin Anticholinergic, decreased ACh activity->decreased tremor |
Sumatriptan | Imitrex triptan |
Eletriptan | Relpax triptan |
Ranitidine | Zantac H2 antag |
Famotidine | Pepcid H2 antag |
Esomeprazole | Nexium PPI |
Lansoprazole | Prevacid PPI |
Omeprazole | Prilosec PPI |
Pantoprazole | Protonix PPI |
Rabeprazole | Aciphex PPI |
Metoclopramide | Reglan dopamine antag->accelerates GI emptying |
Mesalamine | Asacol, Canasa, Lialda, Pentasa, Rowasa inhibits prostaglandin synthesis to inhibit GI inflammation |
Prednisone | Sterapred Corticosteroid |
Methotrexate | Rhematrex Immunosuppressant |
Dexamethasone | Decadron Corticosteroid |
Methylprednisolone | SoluMedrol Corticosteroid |
Codeine | Several Opioid analgesic |
Morphine | Roxanol (liquid), MS Contin, Evinsa, Kadian, Oramorph Narcotic opioid analgesic |
Oxycodone | Oxycontin Opioid analgesic |
Oxycodone/APAP | Percocet Opioid analgesic |
Hydrocodone (in combo only) | With APAP-->Vicodin, Lortab, Lorcet, Anexsia With Ibuprofen-->Vicoprofen |
Citalopram | Celexa SSRI |
Escitalopram | Lexapro SSRI |
Fluoxetine | Prozac, Sarafem, Rapiflux SSRI |
Paroxetine | Paxil SSRI |
Sertraline | Zoloft SSRI |
Amitriptyline | Elavil, Vanatrip TCA |
Nortriptyline | Pamelor, Aventyl TCA |
Duloxetine | Cymbalta SSNRI |
Venlafaxine | Effexor SSNRI |
Bupropion | Wellbutrin SSNDRI |
Mirtazapine | Remeron TetraCA |
Alprazolam | Xanax BZD |
Clonazepam | Klonopin BZD |
Diazepam | Valium BZD |
Lorazepam | Ativan BZD |
Buspirone | Bupsar Anxiolytic |
Venlafaxine | Effexor SNRI |
Hydroxyzine | Vistaril Anxiolytic via H1 receptor |
Lithium | Lithobid |
Olanzepine | Zyprexa AAP |
Ziprasidone | Geodon AAP |
Risperidone | Risperdal AAP |
Tramadol | Ultram |
Etodolac | Acetic acid NSAID |
Indomethacin | Indocin Acetic acid NSAID |
Diclofenac | Cataflam, Voltaren Acetic acid NSAID |
Ibuprofen | Motrin, Advil NSAID |
Naproxen | Naprosyn |
Naproxen sodium | Anaprox NSAID |
Piroxicam | Feldene NSAID more cox 2 selective |
Meloxicam | Mobic NSAID mroe cox 2 selective |
Celecoxib | Celebrex Cox 2 inhibitor |
Hydroxychloroquine | Plaquenil Immunosuppressant like |
Alendronate | Fosamax bisphosphonate |
Risedronate | Actonel bisphosphonate |
Ibandronate | Boniva bisphosphonate |
Raloxifene | Evista SERM |
Cochicine | inhibits lactic acid production to decrease uric acid production |
Allupurinol | Zyloprim xanthine oxidase inhibitor to impair conversion of xanthine oxidase to uric acid |
Probenecid | uricosuric agent to increase renal clearance of uric acid by inhibiting tubular reabsorption |
Nabumetone | Reclafen NSAID |
Propoxyphene/APAP | Darvocet Narcotic analgesic |
Fentanyl | Duragesic, Actiq, Fentora Narcotic analgesic |
Methadone | Dolophine Narcotic analgesic |
Pregabalin | Lyrica induces release of substance P |
Bimatoprost | Lumigan Prostaglandin analog |
Latanoprost | Xalatan Prostaglandin analog |
Travaprost | Travatan Prostaglandin analog |
Cyanocobalamin | Nascobal B12 |
Folic acid(folate) | Apo-Folic |
Tretinion | Retin-A, Renova, Avita |
Adapalene | Differin |
Methotrexate | Antimetabolite |