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Hypnotics/Anxiolytic
Benzos, etc
| Trade | Generic | Class | FDA | off-label | MOA | Dosage | Metabolism |
|---|---|---|---|---|---|---|---|
| Centrax | prazepam | Benz | anx | ETOH withdrawal, Seizures | 30-60 | ||
| Tranxene | clorazepate | Benz | anx, seizures | 4-40 | |||
| Romazicon | flumazenil | Benz | GABA-a receptor antagonist | ||||
| ProSom | estazolam | Benz | Insomnia | 1-2 | |||
| Halcion | triazolam | Benz | Insomnia(ST) | .25-.50 | Pure CYP3A4 substrate | ||
| Xanax | alprazolam | Benz | Panic | Anx | .25-4 | ||
| Rozerem | remelteon | Non-benz hyp | Insomnia | melatonin receptor agaonist | 8 | ||
| Dalmane | flurazepam | Benz | Insomnia(ST) | 15-30 | |||
| Doral | quazepam | Benz | Insomnia (ST) | 7.5-15 | |||
| Ambien | zolpidem | Non-benz hyp | Insom-DFA, SCD(ST) | 5-12.5 | |||
| Sonata | zaleplon | Non-benz hyp | Insomnia (ST) | 5-10 | |||
| Lunesta | eszopiclone | Non-benz hyp | Insomnia (<6 months use) | 2-3 | |||
| BuSpar | buspirone | anti-anxiety | anti-anxiety | inc 5HT,NE, DA | 15-60 | ||
| Klonopin | clonazepam | Benz | Seiz, panic | GAD, hyp | .25-4 | ||
| Restoril | temazepam | Benz | Insomnia (ST) | 15-30 | |||
| Serax | oxazepam | Benz | anx, etoh withdrawal | anti-itch, sez, hyp | 30-120 | ||
| Ativan | lorazepam | Benz | anx | 2-6 | |||
| midazolam | Benz | ||||||
| Librium | chlordiazepoxide | Benz | anx,ETOH withdrawal | 5-100 | |||
| Valium | diazepam | Benz | anx, muscle spasms, seizures | 4-40 | |||
| Baclofen | Benz | GABAb receptor agonist | |||||
| Niravam | alprazolam | Benz | Panic, GAD | .3-5 |