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Interactions
Cyp inhibitors/inducers 1
Question | Answer |
---|---|
CYP 1A2 substrates (some) | theophylline, mexiletine, imipramine, naproxen, propranolol, tracrine, clozapine, cyclobenzapine |
Fluoroquinolones inhibit what in general | inhibit CYP 1A2 |
Fluvoxamine | Inhibit CYP 1A2 |
Cimetidine | Inhibit CYP 1A2, CYP 3A4, CYP 2D6, |
Ticlopidine | Inhibit CYP 1A2 |
CYP 3A substrates (most) | CCBs, Benzos, HIV PI's, HMG - CoA, Cyclosporine, Buspirone, gleevac, haloperidol, pimozide, sildenafil, tamoxifen, trazodone, lapitnibnote classes are general may not be all |
Ketoconazole | inhibit CYP 3A4, CYP 2C19, |
Itraconazole | inhibit CYP 3A4, |
Fluconazole | inhibt 3A4, 2C19 |
Clarithromycin | Inhibit 3A4, |
Erythromycin | Inhibit CYP 3A4, |
Tobacco | induces CYP 1A2 |
Grapefruit juice | Inhibit 3A4, |
Indinavir | Inhibit 3a4., |
Ritinovir | Inhibit 3A4, induces 3A4 |
Nelfinavir | Inhibit 3A4 , |
Nefazodone | Inhibit 3A4, |
Diltiazem | Inhibit 3A4, |
Carbamazepine | Induce 3A4, |
Rifampin | Induce 3A4 |
Rifabutin | Induce 3A4 |
Ritonavir | Induce 3A4 |