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Pharmacology
Final 2008
| Question | Answer |
|---|---|
| clonidine | alpha 2 agonist |
| catapress | alpha 2 agonist |
| methyldopa | *pro drug -alpha 2 agonist |
| guanabenz | alpha 2 agonist |
| guanfacine | alpha 2 agonist |
| dexmedetamidine | alpha 2 agonist |
| brimonidine | alpha 2 agonist *eye |
| alphagan | alpha 2 agonist |
| apraclonidine | alpha 2 agonist |
| yohimbine | alpha 2 ANTagonist |
| labetolol | beta 1,2 and alpha 1 antagonist |
| carvedilol | beta 1, 2 and alpha 1 antagonist |
| coreg | beta 1, 2 and alpha 1 antagonist |
| midodrine | alpha 1 agonist |
| phenylephrine | alpha 1 agonist |
| psuedoephedrine | alpha 1 agonist |
| sudafed | alpha 1 agonist |
| oxymetazolene | alpha 1 agonist |
| afrin | alpha 1 agonist |
| prazosin | alpha 1 antagonist |
| terazosin | alpha 1 antagonist |
| hytrin | alpha 1 antagonist |
| doxazosin | alpha 1 antagonist |
| cardura | alpha 1 antagonist |
| alfuzosin | alpha 1 antagonist |
| oroxatral | alpha 1 antagonist |
| tamsulosin | alpha 1 antagonist *selective to alpha 1a |
| flomax | alpha 1 antagonist *selective to alpha 1a |
| phentolamine | alpha antagonist *non selective |
| phenoxybenzamine | alpha antagonist *non selective *pheochromocytoma |
| albuterol | beta 2 agonist |
| bitolerol | beta 2 agonist |
| formoterol | beta 2 agonist |
| foradil | beta 2 agonist |
| isoethaine | beta 2 agonist |
| levalbuterol | beta 2 agonist |
| metaproternol | beta 2 agonist |
| alupent | beta 2 agonist |
| pirbuterol | beta 2 agonist |
| maxair | beta 2 agonist |
| salmuterol | beta 2 agonist |
| servent | beta 2 agonist |
| terbutaline | beta 2 agonist *used specifically for status asmaticus |
| ritodrine | beta 2 agonist *IV for premature labor |
| isoproterenol | beta agonst *non selective |
| propanolol | beta antagonist *non selective |
| inderal | beta antagonist *non selective |
| nadolol | beta antagonist *non selective |
| pindolol | beta antagonist *non selective |
| sotalol | beta antagonist *non selective |
| timolol | beta antagonist *non selective |
| levobunolol | beta antgonist *non selective |
| dobutamine | beta 1 agonist |
| acebutolol | beta 1 antagonist *partial agonist put in agonist class |
| sectral | beta 1 antagonist *partial agonist put in agonist class |
| atenolol | beta 1 antagonist |
| tenormin | beta 1 antagonist |
| betaxolol | beta 1 antagonist |
| bisoprolol | beta 1 antagonist |
| metoprolol | beta 1 antagonist |
| lopressor | beta 1 antagonist |
| toprolol | beta 1 antgonist |
| esmolol | beta 1 antgonist |
| breuibla | beta 1 antgonist *plasma estraces will decrease T1/2 |
| flolan | sythetic prostacyclin analogs |
| epoprostenol | synthetic prostacyclin analogs |
| ventavis | synthetic prostacyclin analogs |
| iloprost | sythetic prostacyclin analogs |
| treprostinil | synthetic prostacyclin analogs |
| bosentan | endothelian receptor antagonist |
| ambrisentan | endothelian recepter antagonist |
| sildinafil | PDE5 -I |
| revatio | PDE5 -I |
| viagra | PDE5 -I |
| tadinafil | PDE5 -I |
| cialis | PDE5-I |
| vardinafil | PDE5-I |
| levitra | PDE5-I |
| Quinidine | 1a sodium channel blockers |
| procainamide | 1a sodium channel blockers |
| disopyramide | 1a sodium channel blockers |
| lidocaine | 1b sodium channel blockers |
| medilitene | 1b sodium channel blockers |
| flecanide | 1c sodium channel blockers |
| proafenone | 1c sodium channel blockers |
| ibutilide | potassium channeln blockers -class 3 |
| sotalol | potassium channel blockers -class 3 *also beta blocker |
| dofetilide | potassium channel blocker -class 3 |
| amiodarone | potassium channel blocker -dirty drug! also works on Ca+/Na+/and adrenergic recepters! |
| atorvastatin | statin |
| lipitor | statin |
| fluvastatin | statin |
| lesacol | statin |
| mevacor | statin *prodrug |
| luvastatin | statin *prodrug |
| pravastatin | statin |
| pravachol | statin |
| rosuvastatin | statin |
| crestor | statin |
| simvastatin | statin *prodrug |
| zocor | statin *prodrug |
| choestyrine | bile acid sequestrant |
| questran | bile acid sequestrant |
| colestipol | bile acid sequestrant |
| colestid | bile acid sequestrant |
| welchol | bile acid sequestrant |
| zetia | dietary cholesterol uptake inhibitor |
| ezetimibe | dietary cholesterol uptake ihibitor |
| niacin | vitamin b! increases HDL and lowers LDL |
| digoxin | cardiac glycoside |
| adenosine | used rapidily for acute heart failure, get that heart pumping againg |
| manitol | osmotic diuretics |
| urea | osmotic diuretic |
| glycerin | osmotic diuretic |
| AHD | antidiarettic hormone |
| vasopressin | AHD |
| desmopressin DDAVP | works like anti diueretic hormone |
| benazepril | ACEI |
| lotensin | ACE |
| captopril | acei |
| capotin | ACEI |
| Enalopril | ACEI |
| vasotec | ACEI *prodrug |
| enaoloprilat | ACEI |
| fosinopril | acei |
| manopril | ACEI |
| lisinopril | ACEI |
| prinivil | ACEI |
| moexipril | ACEI |
| Univasc | ACEI |
| perindopril | ACEI |
| aceon | ACEI |
| Quinapril | ACEI |
| ramipril | ACEI |
| trandolopril | ACEI |
| mavik | ACEI |
| Alikiren | Renin inhibitor |
| Tekturna | Renin inhibitor |
| canastertan cilexill | ARBS |
| atacand | arb |
| eprosartan | arb |
| teventen | arb |
| irebesartan | arb |
| avapro | arb |
| losartan | arb |
| cozarr | arb |
| olemesartan medoxomel | arb |
| benicar | arb |
| telmisartan | arb |
| valsartan | arb |
| diovan | arb |
| acetazolamide | carbonic anhydrase inhibitor |
| diamox | carbonic anhydase inhibitor |
| methazolamide | carbonic anhydrase inhibitor |
| durzolamide | carbonic anyhrase inhibitor |
| trusopt | carbonic anyhydrous inbitor |
| HCTZ | thiazide like diuretics |
| chlorothaizide | thaizide like diuretics |
| indapamide | thiazide |
| lozal | thiazide |
| metolazone | thiazide |
| zaroxolyn | thiazide |
| furosemide | loop |
| lasix | loop |
| bumetanide | loop |
| bumex | loop |
| toremide | loop |
| ethacrynic acid | loop |
| spirinolactone | potassium sparring diuretic |
| eplerenone | potassium sparring diuretic |
| inspra | potassium sparring diuretic |
| amlodipine | calium channel blocker |
| norvasc | calcium channel blocker |
| felodipine | calcium channel blocker |
| plendil | calcium channel blocker |
| isradipine | calcium channel blocker |
| pynarinic | calcium channel blocker |
| nicardipine | calicium channel blocker |
| cardura | calcium channel blocker |
| nifedipine | calcium channel blocker |
| adalt | calcium channel blocker |
| procardia | calcium channel blocker |
| diltiazem | calcium channel blocker * more selective to the heart |
| cardiazem | calcium channel blocker *more selective to the heart |
| verapamil | calcium channel blocker *more selective to the heart |
| calan | calcium channel blocker *more selective to the heart |
| nimodine | calcium channel blocker |
| nimotop | calcium channel blocker |
| nisoldipine | calcium channel blocker |
| sular | calcium channel blocker |
| sodium nitroprusside | direct acting vasodilator |
| nitroglycerin | direct acting vasodilator |
| hydralazine | direct acting vasodilator |
| bidil | direct acting vasodilator |
| minoxidil | potassium channel blockers *prodrug |
| pinacidil | potassium channel blockers |
| nicarandil | potassium channel blockers |
| crumaklium | potassium channel blockers |
| DIAZOXIDE | potassium optening agent |
| hyperstati | potassium opening agent *arterial vasodilator |
| fenoldopam | dopamine receptor agonist *D1 |
| adderall | amphetamine |
| dexedrine | amphetamine |
| dextriamphetamine | amphetamine |
| desoxyn | amphetamine |
| methamphetamine | amphetamine |
| vyvanse | amphetamine |
| bisdextroamphetamine | amphetamine |
| ritalin | methylphenidate |
| concerta | methylphenidate |
| focalin | methylphenidate |
| dextromethylphenidate | methylphenidate |
| benzphetamine | amphetamine-like anorexants |
| didrex | amphetamine like anorexant |
| diethylpropion | amphetamine like anorexant |
| phendiinetrazine | amphetamine like anorexant |
| Fen-Phen | amphetamine like anorexant |
| meridia | anorexant inhibits seratonin more then NE |
| sibutramine | anorexant inhibits setatonin more then NE |
| provigil | increase wakefullness |
| nuvigil | increase wakefullness |
| modafinil | increase wakefullness |
| cormodafinil | increase wakfulness |
| psuedoephedrine | mixed acting sympathomimetic |
| ephedrine | mixed acting sympathomimetic |
| strattera | increase reuptake of NE |
| succinyl choline | Nicotinic -m- agonist |
| mecamylame | nicotinic -n- antagonist |
| inversine | nicotinic -n- antgonist |
| varenicline | partial nicontic antagonist |
| chantix | partial nicontic antagonist |
| -curonium | nicontinc antagonist |
| -curium | nicontinic antagonist |
| carbachol | muscarinic agonist |
| pilocarpine | muscarinic agonist |
| salogen | muscarinic agonist |
| bethanechol | muscarinic agonist |
| urecholine | muscarinic agonist |
| cevimeline | muscarinic agonist |
| evoxac | muscarinic agonist |
| echothiaphate | ACHEI |
| phosphate iodide | ACHEI |
| neostigmine | ACHEI |
| physiostigmine | ACHEI |
| pyridostigmine | ACHEI |
| echrophrium | ACHEI |
| melatrium | ACHEI |
| Mylelase | ACHEI |
| Atropine | muscarinic antagonist |
| tropicamid | muscarinic antagonist |
| cyclopentolate | muscarinic antgonist |
| cyclogyl | muscarinic antagonist |
| glycopyrolate | muscarinic antagonist |
| mepenzolate | muscarinic antagonist |
| propantheline | muscarinic antagonist |
| clindinium | muscarinic antagonist |
| dicyclomine | muscarinic antagonist |
| bentyl | muscaronic antagonist |
| hyosyamine | muscaronic antagonist |
| levisin | muscaronic antagonist |
| scopalamine | muscaronic antagonist |
| belladonna | muscaronic antagonist |
| ipatropium | muscaronic antagonist |
| atrovent | muscaronic antagonist |
| tiotopium | muscaronic antagonist |
| spiva | muscaronic antagonist |
| tolterodine | muscaronic antagonist |
| detrol | muscaronic antagonist |
| oxybutyin | muscaronic antagonist |
| ditropan | muscaronic antagonist |
| paridenacin | muscarinic antagonist |
| enablex | muscarinic antagonist |
| tropium | muscaronic antagonist |
| sanctura | muscaronic antagonist |
| flavoxate | muscaronic antagonist |
| urispas | muscaronic antagonist |