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ans drugs exam 2
| Question | Answer |
|---|---|
| Adrenergic Agonists | sympathomimetics |
| Phenylephrine * | α-agonist, α1 (direct, selective) Adrenergic Agonists (sympathomimetics |
| Isoproterenol* | β-agonist - β1, β2 (direct, non-selective) Adrenergic Agonists (sympathomimetics |
| Epinephrine* | α1, α2, β1, and β2 agonist (direct, non-selective) Adrenergic Agonists (sympathomimetics |
| Norepinephrine* | α1, α2 , β1 agonist, (direct, non-selective) Adrenergic Agonists (sympathomimetics |
| Dobutamine* | β1 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
| Albuterol* | β2 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
| Metaproterenol* | β2 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
| Terbutaline* | β2 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
| Clonidine | α2 agonist (Direct, selective) Adrenergic Agonists (sympathomimetics |
| Oxymetazoline | α1, α2 (direct, non-selective) Adrenergic Agonists (sympathomimetics |
| Ephedrine | α1, α2, β1, β2, releasing agent (mixed acting) Adrenergic Agonists (sympathomimetics |
| Tyramine* | Releasing agent Adrenergic Agonists (sympathomimetics |
| Amphetamine | Releasing agent Adrenergic Agonists (sympathomimetics |
| Cocaine* | Uptake inhibitor Adrenergic Agonists (sympathomimetics |
| Selegiline | MOA inhibitor Adrenergic Agonists (sympathomimetics |
| Entracapone | COMT inhibitor,Adrenergic Agonists (sympathomimetics |
| Phentolamine* | α-antagonist (nonselective) Adrenergic Antagonists |
| Phenoxybenzamine* | α-antagonist (nonselective) Adrenergic Antagonists |
| Prazosin* | α-antagonist α1 selective Adrenergic Antagonists |
| Tamsulosin* | α-antagonist α1 selective Adrenergic Antagonists |
| Terazosin Doxazosin Alfuzosin Indroramin Urapidil Bunazosin | α-antagonist α1 selective Adrenergic Antagonists |
| Yohimbine* | α-antagonist - α2 selective Adrenergic Antagonists |
| Nadolol* | β-antagonist β1 and β2 non-selective 1st generation, Adrenergic Antagonists |
| Pindolol* | β-antagonist β1 and β2 non-selective 1st generation Adrenergic Antagonists |
| Propranolol* | β-antagonist β1 and β2, Adrenergic Antagonists non-selective 1st generation |
| Timolol* | β-antagonist β1 and β2 non-selective 1st generation Adrenergic Antagonists |
| Penbutolol Sotalol Levobunolol Metipranolol | β-antagonist β1 and β2 non-selective 1st generation Adrenergic Antagonists |
| Acebutolol* | β1 – antagonist selective 2nd generation Adrenergic Antagonists |
| Atenolol* | β1 – antagonist selective 2nd generation Adrenergic Antagonists |
| Metoprolol* | β1 – antagonist selective 2nd generation, Adrenergic Antagonists |
| Bisoprolol Esmolol | β1 – antagonist selective 2nd generation, Adrenergic Antagonists |
| Carteolol* | β- and α antagonist non-selective 3rd generation, Adrenergic Antagonists |
| Carvedilol* | β- and α antagonist non-selective 3rd generation Adrenergic Antagonists |
| Bucindolol Labetalol | β- and α antagonist non-selective 3rd generation, Adrenergic Antagonists |
| Betaxolol Celliprolol Nebivolol | β2-antagonist selective 3rd generation, Adrenergic Antagonists |
| DFP* | Irreversible anti-AchE (organophosphates) |
| Echothiophate* | Irreversible anti-AchE (organophosphates) |
| Soman | Irreversible anti-AchE (organophosphates) |
| Sarin | Irreversible anti-AchE (organophosphates) |
| Parathion --> paraoxon | Irreversible anti-AchE Organophosphate poisonous in insects |
| Neostigmine*(+) | Reversible anti-AchE “carbamates” Slowly reversible |
| Physostigmine* | Reversible anti-AchE “carbamates” Slowly reversible |
| Pyridostigmine*(+) | Reversible anti-AchE “carbamates” Slowly reversible |
| Rivastigmine | Reversible anti-AchE “carbamates” Slowly reversible |
| Edrophonium* | Reversible anti-AchE Rapidly reversible |
| Tacrine* | Reversible anti-AchE Rapidly reversible |
| Donepezil | Reversible anti-AchE Rapidly reversible |
| Galantamine | Reversible anti-AchE Rapidly reversible |
| Atropine | Protects mAchR from excessive stimulation by Ach secondary to anti-AchE poisoning |
| 2-PAM | Restores activity of AchE |
| Tubocuraine* (d-TC) | Non-depolarizing neuromuscular blocker |
| Pancuronium* | Non-depolarizing neuromuscular blocker |
| Succinylcholine* | Depolarizing neuromuscular blocker |
| Decamethonium | Depolarizing neuromuscular blocker |
| Na-Dantrolene | Skeletal muscle relaxor used to treat Malignant hyperthermia caused by Succinylcholine |
| Choline | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
| Acetylcholine | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
| Carbamylcholine | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
| Methacholine | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
| Bethanechol | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
| Muscarine | Direct-Acting Muscarinic Receptor Agonists Cholinomimetic Alkaloids /Synthetics Cholinergic Agonists |
| Pilocarpine | Direct-Acting Muscarinic Receptor Agonists Cholinomimetic Alkaloids /Synthetics Cholinergic Agonists |
| Nicotine | Nicotinic agonist Cholinergic Agonists |
| Atropine | Parasympatholytics Belladonna Alkaloids Muscarinic Receptor Antagonists (Cholinolytics) |
| Scopolamine | Parasympatholytics Belladonna Alkaloids Muscarinic Receptor Antagonists (Cholinolytics) |
| Propantheline Glycopyrrolate Pirenzepine Dicyclomine Tropicamide Ipratropium Benztropine | Parasympatholytics Other muscarinic alkaloids Muscarinic Receptor Antagonists (Cholinolytics) |
| Oxybutynin | Anti-cholinergic for overactive bladder Muscarinic Receptor Antagonists (Cholinolytics) |
| Darifenacin | Anti-cholinergic for overactive bladder Muscarinic Receptor Antagonists (Cholinolytics) |
| Tolterodine | Anti-cholinergic for overactive bladder Muscarinic Receptor Antagonists (Cholinolytics) |
| Methoctramine Dramamine Amitriptyline Imipramine Promethazine Chlorpheneramine Diphenhydramine | Anti-muscarinic drugs Muscarinic Receptor Antagonists (Cholinolytics) |