Brand | Generic | Side effects | Drug interactions |
Retrovir | Zidovudine (AZT) | N&V, HA, myalgia, anemia, Mitochondrial. Lipoatrophy | No d4T, ddI. Avoid ganciclovir, interferon, chemo. |
Videx | Didanosine (ddI) | Pancreatitis, Peripheral Neuropathy, N&V Fatigue, Myalgia, Bone Marrow, Mitochondrial, Lipoatrophy | Tenofovir. Decrease dose. No AZT, ddI, d4T |
Zerit | Stavudine (D4T) | Pancreatitis, Peripheral Neuropathy, N&V Fatigue, Myalgia, Bone Marrow, Mitochondrial, Lipoatrophy | No AZT, ddI |
Epivir | Lamivudine (3TC) | Pancreatitis, Liver | |
Ziagen | Abacavir | Hypersensitivity. (fever, rash, GI, Constitutional, Respiratory | |
Emtriva | Emtricitabine | Nausea, rash, diarrhea, HA Black skin dots | |
Viread | Tenofovir | Renal, Liver, GI | Decrease ddI, Boost Atazanavir. |
Sustiva | Efavirenz | Mental status, worsen depression, dreams, hung over, Manic, Rash, DI, Prego D | CYP3A4-mixed No Midazolam, triazolam. causes decreased Methadone. Posa, vori, itra |
Rescriptor | Delaviridine | Rash, Itching, DI, Liver | CYP3A4 Inhibitor |
Edurant | Rilpivirine | Rash, Depression, Insomnia, HA With regular meal | PPIs, H2, antacids, Carbamazepine, phenobarb, phenytoin, dex, Rifampin |
Intelence | Etravirine | Take with food, PG:B, has activity against virus resistant | No Carbamazepine, Phenobarbital, Phenytoin, Rifampin |
Combivir | Zidovudine and Lamivudine | | |
Epzicom | Abacavir and Lamivudine | | |
Truvada | Tenofovir and Emtricitabine | | |
Trizivir | Abacavir, Lamivudine, and Zidovudine | | |
Atripla | Efavirenz, Tenofovir, and Emtricitabine | | |
Complera | Rilpivirine, Tenofovir, and Emtricitabine | | |
Stribild | Elvitegravir, cobicistat, tenofovir, and Emtricitabine | | Cobicistat-CYP3A4 Inhibitor No rifampin |
Invirase | Saquinavir | Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liver | |
Norvir | Ritonavir | N&V, rash, liver DI, circumoral Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liverparesthesias. | CYP3A4 Inhibitor Vori, itra |
Crixivan | Indinavir | Jaundice, stones, skin changes. Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liver | |
Viracept | Nelfinavir | Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liver | |
Lexiva | Fosamprenavir | Rash. Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liver | |
Kaletra | Lopinavir/Ritonavir | Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liver | |
Reyataz | Atazanavir | Hyperbilirubinemia, jaundice, rash, bloating/gas, lipodystrophy(Not as bad as others), increased PR interval. | No PPI, separate H2 by 12 hrs, 2hrs for antacids. No Aaltegravir |
Aptivus | Tipranavir | Liver, CNS bleeding, rash. Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liver | CYP3A4-Inducer |
Prezista | Darunavir | Gas/Bloating, Diarrhea, Nausea, Dry Skin, blood Sugar, Lipids, Lipodystrophy, Osteonecrosis, Liver | |
Fuzeon | Enfuvirtide | Injection site reactions | |
Selzentry | Maraviroc | Hepatotoxicity(BBW), Allergy, Rash, Cough, Sleep | Carbamazepine, phenobarb, Phenytoin, clarithromycin, St. Johns, Vori, Rifabutin, Rifampin |
Isentress | Raltegravir | GI | No Atazanavir, No Rifampin |
Stribild | Elvitegravir, cobicistat, tenofovir, emtricitabine | Nausea, diarrhea, gas, increased Scr | Alfuzocin, sildenafil, cisapride, pimozide, ergots, triazolam, midazolam, simvastatin, lovastatin, rifampin, St. Johns |
Viramune | Nevirapine | Rash, Itching, DI, Liver(BBW) Men CD4>400, Women CD4>250 | CYP3A4 Inducer |