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CNS Drugs
Sleep + Dementia
| Term | Definition |
|---|---|
| Modafanil | Weak DAT inhibition; DAT > NET |
| GHB | Increases dopaminergic disinhibition, decrease GABA |
| Solriamfetol | DA + NE reuptake inhibitor |
| Pitolisant | H3 inverse agonist/antagonist |
| H3 Autoreceptors | Pitolisant increases histamine |
| H3 Heteroreceptors | Pitolisant increases monoamines |
| NBRA | Positive allosteric modulator of GABA-A receptor containing a1 subunits |
| Ramelteon | Selective melatonin agonist; MT1> MT2 |
| Gabapentin | Decreases calcium influx on presynaptic neurons, decreases glutamate |