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Pain/Heme/Onc 1
Pain, Hematology, and Oncology 1
| Generic | Brand | Pharmacologic Category | Common Indications | Key Side Effects | BBW | Other Notes |
|---|---|---|---|---|---|---|
| methadone (PO, IV) | Dolophine | Opioid analgesic | Opioid use disorder, severe chronic pain | Qtc prolongation, dizziness, drowsiness, nausea, vomiting, constipation, respiratory depression (dose-related) | QTc interval prolongation and serious arrhythmia (Torsades de Pointes) have occurred during treatment; concomitant use with CYP3A4, 2B6, 2C19, or 2D6 (or stopping the same inducers) can increase methadone concentrations + All Opioid Analgesics BBWs | |
| fentanyl (transdermal, IV) | Transdermal: Duragesic IV: Sublimaze | Opioid analgesic | Pain | dizziness, drowsiness, itching, nausea, vomiting, constipation, respiratory depression (dose-related) | Opioid addiction/ abuse/misuse/Overdose/death/resp. depression;Pregnancy use:Neonatal opioid withdrawal synd.;Abrupt discont.:Opioid-induced withdrawal synd.;Use w benzo/CNS depres./alcohol:Sedation,resp. depres.,coma, death | |
| hydromorphone (PO, IV) | Dilaudid | Opioid analgesic | Pain | dizziness, drowsiness, itching, nausea, vomiting, constipation, respiratory depression (dose-related) | Opioid addiction/ abuse/misuse/Overdose/death/resp. depression;Pregnancy use:Neonatal opioid withdrawal synd.;Abrupt discont.:Opioid-induced withdrawal synd.;Use w benzo/CNS depres./alcohol:Sedation,resp. depres.,coma, death | |
| morphine (extended release) (PO) | MS Contin, Kadian | Opioid analgesic | Pain | dizziness, drowsiness, itching, nausea, vomiting, constipation, respiratory depression (dose-related) | Opioid addiction/ abuse/misuse/Overdose/death/resp. depression;Pregnancy use:Neonatal opioid withdrawal synd.;Abrupt discont.:Opioid-induced withdrawal synd.;Use w benzo/CNS depres./alcohol:Sedation,resp. depres.,coma, death | |
| morphine (immediate release) (PO, IV, IM, PR) | IV: Duramorph, Infumorph | Opioid analgesic | Pain | dizziness, drowsiness, itching, nausea, vomiting, constipation, respiratory depression (dose-related) | Opioid addiction/ abuse/misuse/Overdose/death/resp. depression;Pregnancy use:Neonatal opioid withdrawal synd.;Abrupt discont.:Opioid-induced withdrawal synd.;Use w benzo/CNS depres./alcohol:Sedation,resp. depres.,coma, death | |
| oxycodone (PO) | Oxycontin, Roxicodone | Opioid analgesic | Pain | dizziness, drowsiness, itching, nausea, vomiting, constipation, respiratory depression (dose-related) | Opioid addiction/ abuse/misuse/Overdose/death/resp. depression;Pregnancy use:Neonatal opioid withdrawal synd.;Abrupt discont.:Opioid-induced withdrawal synd.;Use w benzo/CNS depres./alcohol:Sedation,resp. depres.,coma, death | |
| tramadol (PO) | Ultram, Ultram ER | Central analgesic; partial opioid agonist | Pain | dizziness, drowsiness, nausea, vomiting, constipation, respiratory depression (dose-related) | serious or fatal respiratory depression may occur | lowers seizure threshold |
| acetaminophen (PO, PR, IV) * | PO/PR: Tylenol IV: Ofirmev | Analgesic (non-opioid), antipyretic | Pain, fever | nausea, vomiting, increased hepatic transaminases | total daily dose from all sources should not exceed maximum daily limit; hepatotoxicity |