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Phar - Hague 3
Angina, Vasodilators, CHF
Question | Answer |
---|---|
Beta-blockers | Propanolol Atenolol |
Propranolol properties | non selective beta-adrenergic receptor antagonist Oral |
Propanolol use / side effects | Use -CHF -Hypertension -Angina Side effects -Nausea -Hypotension |
Atenolol properties | selective beta1-adrenergic receptor antagonist Oral |
Atenolol use / side effects | Use -CHF -Hypertension -Angina Side effects -Nausea -Hypotension |
Vasodilators | Nitroglycerine Isosorbide dinitrate |
Nitroglycerine properties | Donate NO, increase cGMP in SMC, PKG activity, vasodilation Oral |
Nitroglycerine use / side effects | Use -Acute decompensated HF -Angina Side effects -Hypotension -Tachycardia |
Isosorbide dinitrate properties | Donate NO, increase cGMP in SMC, PKG activity, vasodilation Oral |
Isosorbide dinitrate use / side effects | Use -Acute decompensated HF -Angina Side effects -Hypotension -Tachycardia |
PDE Inhibitors | Sildenafil |
Sildenafil properties | Inhibitor of cGMP phosphodiesterase Oral |
Sildenafil use / side effects | Use -ED -BPH -Pulmonary hypertension Side effects -Hypotension -Vision |
Ca2+ channel antagonists | Verapamil Diltiazem Nifedipine |
Verapamil properties | Voltage gated Ca channel inhibitor, cardiac/VSM Oral |
Verapamil use / side effects | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |
Diltiazem properties | Voltage gated Ca channel inhibitor, cardiac/VSM Oral |
Diltiazem use / side effects | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |
Nifedipine properties | Voltage gated Ca channel inhibitor, VSM only Oral |
Nifedipine use / side effects | Use -Angina -Hypertension Side effects -Hypotension -Tachycardia |