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Anticholinergic
Term | Definition |
---|---|
Tolterodine (DETROL) Tiotrop[ium] (SPIRIVA) Soli[fenacin] (VESICARE) Dari[fenacin] (ENABLEX) | Muscarinic Antagonist MOA: Blocks Ach at M3 receptors High Dose - May Block other type of Muscarinic Receptors |
Ipratrop[ium] (ATROVENT) Oxtrop[ium] Bromide (OXIVENT) | Muscarinic Antagonist INDC: Asthma / COPD Short Acting Muscarinic Antagonist (SAMAs) |
Tiotrop[ium] (SPIRIVA) Aclidin[ium] Bromide (TUDORZA PRESSAIR) Glycopyrron[ium] Bromide (SEEBRI NEOHALER) Umeclindn[ium] (ELLIPTA) Reve[fenacin] (YUPELRI) | Muscarinic Antagonist INDC: Asthma / COPD Long Acting MAS |
Dicyclomine (BENTYL) Hyoscyamine (LEVSIN) Mebeverine (COLOFAC) | Muscarinic Antagonist INDC: GI Hypermotility IBS-D(iarrhea) |
Homatropine (ISOPTO, HOMATROPINE) - LONG Cyclopentolate (CYCLOGYL) Tropicamide (MYDRIACYL) - SHORT Atropine | Muscarinic Antagonist INDC: Induce Mydriasis MOA: Blocks ACh on eye fibers iris ADR: Inhibitor Overdose, Organophosphate |
Scopolamine (MALDEMAR, SCOPACE) | Muscarinic Antagonist INDC: Motion Sickness MOA: Blocks ACh from activating |
Benztropine (COGENTIN) Trihexyphenidyl (ARTANE) | Muscarinic Antagonist INDC: Parkinson's Disease MOA: Blockage of CNS Musc. Receptors, Reduces Hyperactivity of ACh pathway |
Oxybutynin (DITROPAN) Tolterodine (DETROL) Trospium (SANCTURA) Solifenacin (VESICARE) Darifenacin (ENABLEX) | Muscarinic Antagonist INDC: Urinary Incontinence MOA: Blocks Effects of ACh on M3 receptor |
Glycopyrronium (QBREXZA) | Muscarinic Antagonist INDC: LAMA for excessive sweating MOA: Reduce ACh on sweat Glands ADR: Dry Mouth, Mydriasis, Urinary Hesitation , Blurred Vision, Constipation |
BOTULINUM TOXIN Onabotulinum Toxin A (BOTOX) Abobotulinum Toxin A (DYSPORT) Rimabotulinum Toxin B (MYOBLOC) | Muscarinic Antagonist INDC: Anti wrinkling, hyperhidrosis, skeletal muscle, spasticity, migraine MOA: DEC ACh release from cholinergic nerve by irreversibly binding to neuromuscular junction ADR: Fatal Neuroparalytic illness by bacterium |