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ans drugs exam 2
Question | Answer |
---|---|
Adrenergic Agonists | sympathomimetics |
Phenylephrine * | α-agonist, α1 (direct, selective) Adrenergic Agonists (sympathomimetics |
Isoproterenol* | β-agonist - β1, β2 (direct, non-selective) Adrenergic Agonists (sympathomimetics |
Epinephrine* | α1, α2, β1, and β2 agonist (direct, non-selective) Adrenergic Agonists (sympathomimetics |
Norepinephrine* | α1, α2 , β1 agonist, (direct, non-selective) Adrenergic Agonists (sympathomimetics |
Dobutamine* | β1 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
Albuterol* | β2 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
Metaproterenol* | β2 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
Terbutaline* | β2 agonist (direct, selective) Adrenergic Agonists (sympathomimetics |
Clonidine | α2 agonist (Direct, selective) Adrenergic Agonists (sympathomimetics |
Oxymetazoline | α1, α2 (direct, non-selective) Adrenergic Agonists (sympathomimetics |
Ephedrine | α1, α2, β1, β2, releasing agent (mixed acting) Adrenergic Agonists (sympathomimetics |
Tyramine* | Releasing agent Adrenergic Agonists (sympathomimetics |
Amphetamine | Releasing agent Adrenergic Agonists (sympathomimetics |
Cocaine* | Uptake inhibitor Adrenergic Agonists (sympathomimetics |
Selegiline | MOA inhibitor Adrenergic Agonists (sympathomimetics |
Entracapone | COMT inhibitor,Adrenergic Agonists (sympathomimetics |
Phentolamine* | α-antagonist (nonselective) Adrenergic Antagonists |
Phenoxybenzamine* | α-antagonist (nonselective) Adrenergic Antagonists |
Prazosin* | α-antagonist α1 selective Adrenergic Antagonists |
Tamsulosin* | α-antagonist α1 selective Adrenergic Antagonists |
Terazosin Doxazosin Alfuzosin Indroramin Urapidil Bunazosin | α-antagonist α1 selective Adrenergic Antagonists |
Yohimbine* | α-antagonist - α2 selective Adrenergic Antagonists |
Nadolol* | β-antagonist β1 and β2 non-selective 1st generation, Adrenergic Antagonists |
Pindolol* | β-antagonist β1 and β2 non-selective 1st generation Adrenergic Antagonists |
Propranolol* | β-antagonist β1 and β2, Adrenergic Antagonists non-selective 1st generation |
Timolol* | β-antagonist β1 and β2 non-selective 1st generation Adrenergic Antagonists |
Penbutolol Sotalol Levobunolol Metipranolol | β-antagonist β1 and β2 non-selective 1st generation Adrenergic Antagonists |
Acebutolol* | β1 – antagonist selective 2nd generation Adrenergic Antagonists |
Atenolol* | β1 – antagonist selective 2nd generation Adrenergic Antagonists |
Metoprolol* | β1 – antagonist selective 2nd generation, Adrenergic Antagonists |
Bisoprolol Esmolol | β1 – antagonist selective 2nd generation, Adrenergic Antagonists |
Carteolol* | β- and α antagonist non-selective 3rd generation, Adrenergic Antagonists |
Carvedilol* | β- and α antagonist non-selective 3rd generation Adrenergic Antagonists |
Bucindolol Labetalol | β- and α antagonist non-selective 3rd generation, Adrenergic Antagonists |
Betaxolol Celliprolol Nebivolol | β2-antagonist selective 3rd generation, Adrenergic Antagonists |
DFP* | Irreversible anti-AchE (organophosphates) |
Echothiophate* | Irreversible anti-AchE (organophosphates) |
Soman | Irreversible anti-AchE (organophosphates) |
Sarin | Irreversible anti-AchE (organophosphates) |
Parathion --> paraoxon | Irreversible anti-AchE Organophosphate poisonous in insects |
Neostigmine*(+) | Reversible anti-AchE “carbamates” Slowly reversible |
Physostigmine* | Reversible anti-AchE “carbamates” Slowly reversible |
Pyridostigmine*(+) | Reversible anti-AchE “carbamates” Slowly reversible |
Rivastigmine | Reversible anti-AchE “carbamates” Slowly reversible |
Edrophonium* | Reversible anti-AchE Rapidly reversible |
Tacrine* | Reversible anti-AchE Rapidly reversible |
Donepezil | Reversible anti-AchE Rapidly reversible |
Galantamine | Reversible anti-AchE Rapidly reversible |
Atropine | Protects mAchR from excessive stimulation by Ach secondary to anti-AchE poisoning |
2-PAM | Restores activity of AchE |
Tubocuraine* (d-TC) | Non-depolarizing neuromuscular blocker |
Pancuronium* | Non-depolarizing neuromuscular blocker |
Succinylcholine* | Depolarizing neuromuscular blocker |
Decamethonium | Depolarizing neuromuscular blocker |
Na-Dantrolene | Skeletal muscle relaxor used to treat Malignant hyperthermia caused by Succinylcholine |
Choline | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
Acetylcholine | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
Carbamylcholine | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
Methacholine | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
Bethanechol | Direct-Acting Muscarinic Receptor Agonists Choline Esters Cholinergic Agonists |
Muscarine | Direct-Acting Muscarinic Receptor Agonists Cholinomimetic Alkaloids /Synthetics Cholinergic Agonists |
Pilocarpine | Direct-Acting Muscarinic Receptor Agonists Cholinomimetic Alkaloids /Synthetics Cholinergic Agonists |
Nicotine | Nicotinic agonist Cholinergic Agonists |
Atropine | Parasympatholytics Belladonna Alkaloids Muscarinic Receptor Antagonists (Cholinolytics) |
Scopolamine | Parasympatholytics Belladonna Alkaloids Muscarinic Receptor Antagonists (Cholinolytics) |
Propantheline Glycopyrrolate Pirenzepine Dicyclomine Tropicamide Ipratropium Benztropine | Parasympatholytics Other muscarinic alkaloids Muscarinic Receptor Antagonists (Cholinolytics) |
Oxybutynin | Anti-cholinergic for overactive bladder Muscarinic Receptor Antagonists (Cholinolytics) |
Darifenacin | Anti-cholinergic for overactive bladder Muscarinic Receptor Antagonists (Cholinolytics) |
Tolterodine | Anti-cholinergic for overactive bladder Muscarinic Receptor Antagonists (Cholinolytics) |
Methoctramine Dramamine Amitriptyline Imipramine Promethazine Chlorpheneramine Diphenhydramine | Anti-muscarinic drugs Muscarinic Receptor Antagonists (Cholinolytics) |