First Aid - Pharm 3

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Cholinomimetics;direct;names   Bethanechol ;Carbachol ;Pilocarpine ;Methacholine  
Cholinomimetics;indirect;names   Neostigmine ;Pyridostigmine ;Edrophonium ;Physostigmine ;Echothiophate  
Bethanechol ;;Mech   Cholinomimetics: Direct agonist  
Carbachol ;;Mech   Cholinomimetics: Direct agonist  
Pilocarpine ;;Mech   Cholinomimetics: Direct agonist  
Methacholine ;;Mech   Cholinomimetics: Direct agonist  
Neostigmine ;;Mech   Cholinomimetics: inirect agonist (anticholinesterase);;↑ endogenous ACh  
Pyridostigmine ;;Mech   Cholinomimetics: inirect agonist (anticholinesterase);;↑ endogenous ACh  
Edrophonium ;;Mech   Cholinomimetics: inirect agonist (anticholinesterase);;↑ endogenous ACh  
Physostigmine ;;Mech   Cholinomimetics: inirect agonist (anticholinesterase);;↑ endogenous ACh  
Echothiophate ;;Mech   Cholinomimetics: inirect agonist (anticholinesterase);;↑ endogenous ACh  
Which Cholinergic Activates Bowel and Bladder smooth muscle;   Bethanechol  
Which Cholinergic Contracts ciliary muscle of eye (open angle), pupillary sphincter (narrow angle)   Carbachol  
Which Cholinergic Stimulates muscarinic receptors in airway when inhaled.   Methacholine  
Which Cholinergic ;;Potent stimulator of sweat, tears, saliva   Pilocarpine  
Which Cholinergic resistant to AChE   Bethanechol and Pilocarpine  
Which Cholinergic ↑ endogenous ACh No CNS penetration   Neostigmine  
Which Cholinergic ↑ endogenous ACh; ↑ strength   Pyridostigmine  
Which Cholinergic is used for Postoperative and neurogenic ileus and urinary ;retention   Bethanechol ;and;Neostigmine  
Which Cholinergic is used for Glaucoma, pupillary contraction, and release of intraocular pressure   Carbachol, Echothiophate and Physostigmine  
Which Cholinergic is used for Potent stimulator of sweat, tears, saliva   Pilocarpine  
Which Cholinergic is used for Challenge test for diagnosis of asthma   Methacholine  
Which Cholinergic is used for reversal of ;neuromuscular junction blockade (postoperative)   Neostigmine  
Which Cholinergic is used for Myasthenia gravis   Neostigmine ;;Pyridostigmine does penetrate CNS  
Which Cholinergic is used for Diagnosis of myasthenia gravis   Edrophonium  
Which Cholinergic is used for atropine overdose   Physostigmine  
Clinical applications of;;Bethanechol   Postoperative and neurogenic ileus and urinary ;retention  
Clinical applications of;;Carbachol   Glaucoma, pupillary contraction, and release of ;intraocular pressure  
Clinical applications of;;Pilocarpine   Potent stimulator of sweat, tears, saliva  
Clinical applications of;;Methacholine   Challenge test for diagnosis of asthma  
Clinical applications of;;Neostigmine   Postoperative and neurogenic ileus and urinary ;retention, myasthenia gravis, reversal of ;neuromuscular junction blockade (postoperative)  
Clinical applications of;;Pyridostigmine   Myasthenia gravis; does penetrate CNS  
Clinical applications of;;Edrophonium   Diagnosis of myasthenia gravis (extremely short ;acting)  
Clinical applications of;;Physostigmine   Glaucoma (crosses blood-brain barrier → CNS) ;and atropine overdose  
Clinical applications of;;Echothiophate   Glaucoma  


   

 
 

 
 

 

 

 
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