Question | Answer |
Cimetidine trade name | Tagamet |
Cimetidine class | H2 antag |
Ranitidine trade name | Zantac |
Ranitidine class | H2 antag |
Famotidine trade name | Pepcid |
Famotidine class | H2 antag |
Omeprazole trade name | Prilosec |
Omeprazole class | Proton pump inhibitor |
Metronidazole class | Nitroimidazol antibiotic |
Amoxicillin class | Penicillin antibiotic |
Clarithomycin class | Macrolide antibiotic |
AlOH3 and MgOH2 trade name | Mylanta, Maalox |
Mylanta, Maalox class | Antacid Salt |
Calcium Carbonate trade name | Tums |
Tums class | Antacid Salt |
Sodium Bicarbonate trade name | Alka Seltzer |
Alka Seltzer class | Antacid Salt |
Sucralfate trade name | Carafate |
Sucralfate class | Mucosal protective agent |
Misoprostol trade name | Cytotec |
Misoprostol class | Mucosal Protective Agent |
Bismuth Subasalicylate trade name | Pepto Bismol |
Bismuth Subsalicylate class | Mucosal Protective Agent |
Metoclopramide trade name | Reglan |
Metoclopramide class | Prokinetic Agent |
Cimetadine Adverse | blocks P450s |
Famotidine Advantage | does not inhibit first pass ethanol metabolism |
Proton Pump Inhibitor MOA | covalent modification of H/K ATPase- irreversible |
Zollinger-Ellison treatment of choice | Proton Pump Inhibitors |
Sucralfate MOA | produces protective covering of ulceration |
Misoprostol MOA | Prostaglandin receptor agonist- inc. secretion of mucous and bicarb |
Misoprostol Adverse | causes myometrial contrxn- no use in pregnancy |
Metoclopramide MOA | 5-HT4 receptor agonist- gastric emptying |
Ciprofloxacin trade name | Cipro |
Ciprofloxacin class | Fluorinated 4-quinolone |
Ofloxacin trade name | Floxin |
Ofloxacin class | Fluorinated 4-quinolone |
Norfloxacin class | Fluorinated 4-quinolone |
Octreotide trade name | Sandostatin |
Octreotide class | Somatostatin analog |
Diphenoxylate trade name | Lomotil |
Diphenoxylate class | Piperidine opioid mu agonist |
Difenoxin trade name | Motofen |
Difenoxin class | Piperidine opioid mu agonist |
Loperamide trade name | Imodium |
Loperamide class | Piperidine opioid mu agonist |
Ondensatron trade name | Zofran |
Ondensatron class | 5-HT3 Antagonist |
Granisetron trade name | Kytril |
Granisetron class | 5-HT3 Antagonist |
Trimethobenzamide trade name | Tigan |
Trimethobenzamide class | D2 antagonist- prokinetic agent |
Chlorpromazine trade name | Thorazine |
Chlorpromazine class | Neuroleptic |
Prochlorperazine trade name | Compazine |
Prochlorperazine class | Neuroleptic |
Heloperidol trade name | Haldol |
Heloperidol class | Neuroleptic |
Dexamethasone class | Glucocorticoid |
Dronabinol trade name | Marinol (pot) |
Dronabinol class | Cannabinoid |
Lorazepam trade name | Ativan |
Lorazepam class | Benzodiazepines |
Promethazine class | Antihistamine |
Scopolamine class | Anticholinergic |
Ipecac | Emetic |
Opioid MOA | Reduced motility, acid- antidiarrheal |
Fluorinated 4- quinolones MOA | Inhibit A subunit of DNA gyrase |
Bismuth salicylate MOA | coating ulceration (dyspepsia), antimicrobial(ulcers and diarrhea) |
mu opioid agonists MOA | inhib of presynaptic nerves of myenteric plexus- low motility |
Difenoxylate, Difenoxin Adverse | Affect CNA- can be addictive |
Octreotide MOA | Interaction with somatostatin receptor |
Octreotide Adverse | gallstones due to decreased emptying |
5-HT3 receptor antagonists MOA | block 5-HT3 receptor- anti-emetics |
Metoclopramide anti-emetic MOA | 5-HT3 agonist, D2 antag- inc. motility |
Dexamethasone MOA | decrease inflammation- anti-emetic |
Dronabinol MOA | Cannabinoid agonist- anti-emetic |
Promethazine, Diphenylhydramine MOA | H1 receptor antagonists- motion sickness and vertigo |
Scopolamine MOA | Muscarinic antagonist- motion sickness |
Apomorphine class | pro-emetic (poisoning)- stimulates the CTZ |
Diuretics | Compounds that produce salt excretion |
Diuretic uses | CHF, Hypertension, Edema |
Acetazolamide trade name | Diamox |
Acetazolamide class | CA inhibitor |
Dichlorophenamide trade name | Daranide |
Dichlorophenamide class | CA inhibitor |
Methazolamide trade name | Neptazane |
Methazolamide class | CA inhibitor |
CA inhibitor uses | Glaucoma, Cerebral Edema, Alkalosis |
CA inhibitor MOA | dec. reabs. of bicarb |
Glycerin class | Osmotic Diuretic |
Isosorbide class | Osmotic Diuretic |
Mannitol class | Osmotic Diuretic |
Urea class | Osmotic Diuretic |
Osmotic Diuretic MOA | osmotically keep water in tubule- excretion |
Ethacrynic Acid trade name | Edecrin |
Ethacrynic Acid class | Loop Diuretic |
Furosemide trade name | Lasix |
Furosemide class | Loop Diuretic |
Bumetanide trade name | Bumex |
Bumetanide class | Loop Diuretic |
Torsemide trade name | Demadex |
Torsemide class | Loop Diuretic |
Loop Diuretic MOA | look up! |
Loop Diuretic secretion | not filtered- secreted in prox tubule |
Loop Diuretic adverse | K+ wasting, hyponatremia |
Chlorothiazide trade name | Diuril |
Chlorothiazide class | Thiazide diuretic |
Hydrochlorothiazide trade name | Hydrodiuril |
Hydrochlorothiazide class | Thiazide diuretic |
Thiazide MOA | Inhib NaCl symport in dist tubule |
Thiazide adverse | tolerance after 1 wk, lethal with Quinidine (antiarrhythmetic) |
Amiloride trade name | Midamor |
Triamterene trade name | Dyrenium, Maxide |
Amiloride class | Na+ channel inhibitor |
Triamterene class | Na+ channel inhibitor |
Na+ channel inhib advantage | K+ sparing |
Na+ channel inhib MOA | Inhib Na+ channel in dist tubule |
Spironolactone trade name | Aldactone |
Spironolactone class | Aldosterone Antagonist |
Aldosterone Antagonist MOA | Prevents ALDO-MR binding, dec. Na+ reabs and K+ secretion |
T. enanthate, cypionate, propionate | IM Testosterone replacements |
Testoderm | Transcrotal Testosterone replacement |
Androderm | Transdermal Testosterone replacement patch |
Androgel | Transdermal Testosterone replacement gel |
Testopel | subQ implant testosterone replacement |
Sildenafil trade name | Viagra |
Sildenafil MOA | PDE 5 inhibitor- inc. cGMP, vasodilation |
Sildenafil use | Tx. of ED |
Vardenafil trade name | Levitra |
Vardenafil MOA | PDE 5 inhibitor- inc. cGMP, vasodilation |
Vardenafil use | Tx. of ED |
Tadalafil trade name | Cialis |
Tadalafil MOA | PDE 5 inhibitor- inc. cGMP, vasodilation |
Tadalafil use | Tx. ED |
Yohimbine class | a2 adrenergic antagonist |
Yohimbine use | Tx. psychogenic ED |
Papaverine | opioid peptide |
Papaverine | injected tx. for ED |
Phentolamine | alpha adrenergic antag |
Phentolamine | injected tx. for ED |
Alprostadil class | PGE1 |
Alprostadil admin route | penile injection or urethral pellet |
Alprostadil use | Tx. ED |